| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5278465 | 33 | IC50 | > | 2 | uM | ALA5252878 | nM | Homo sapiens | |||
| 2. |  ALA3586447 | 11 | INH | = | 83 | % | ALA5252735 | % | Homo sapiens | |||
| 3. |  ALA3586443 | 7 | INH | = | 15 | % | ALA5252735 | % | Homo sapiens | |||
| 4. |  4-Aminocinnoline-3-carboxamide | HTS-9026 | INH | = | 90.1 | % | ALA5252735 | % | Homo sapiens | |||
| 5. | 4-Aminocinnoline-3-carboxamide | HTS-9026 | Kd | > | 10000 | nM | ALA5252716 | nM | Homo sapiens | |||
| 6. |  ALA5270781 | 38 | IC50 | > | 2 | uM | ALA5252051 | nM | Homo sapiens | |||
| 7. |  ALA3932338 | BDBM250054 | IC50 | = | 1.3 | nM | ALA5251918 | 8.89 | nM | Homo sapiens | ||
| 8. |  ALA5276374 | (S)-20a; BGB-8035 | IC50 | = | 15 | nM | ALA5251918 | 7.82 | nM | Homo sapiens | ||
| 9. |  ALA4560385 | 9a | IC50 | = | 0.9 | nM | ALA5243498 | 9.05 | nM | Homo sapiens | ||
| 10. |  mobocertinib | MOBOCERTINIB | INH | > | 81 | % | ALA5238875 | % | Homo sapiens | |||
| 11. |  Selitrectinib (LOXO-195) | SELITRECTINIB | % of control | = | 15 | % | ALA5213060 | % | Homo sapiens | |||
| 12. |  ALA4577237 | EUB0000549 | % of control | = | 40 | % | ALA5214576 | % | Homo sapiens | |||
| 13. |  BAY-293 | EUB0000320 | % of control | = | 49 | % | ALA5213884 | % | Homo sapiens | |||
| 14. |  Acalabrutinib (ACP-196) | ACALABRUTINIB | IC50 | = | 46 | nM | ALA5213056 | 7.34 | nM | Homo sapiens | ||
| 15. |  Zanubrutinib (BGB-3111) | BDBM250082 | IC50 | = | 0.62 | nM | ALA5210356 | 9.21 | nM | Homo sapiens | ||
| 16. | Zanubrutinib (BGB-3111) | BDBM250082 | IC50 | = | 360 | nM | ALA5209941 | 6.44 | nM | Homo sapiens | ||
| 17. |  BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 0.07 | C | ALA5209691 | C | Homo sapiens | |||
| 18. |  Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.84 | C | ALA5209691 | C | Homo sapiens | |||
| 19. |  AZD6482 | AZD-6482 | Delta TM | = | 0.05 | C | ALA5209691 | C | Homo sapiens | |||
| 20. |  ASP3026 | ASP-3026 | Delta TM | = | 2.72 | C | ALA5209691 | C | Homo sapiens |
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