# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA519881 | 15h | INH | = | 7 | % | ALA5252730 | % | Homo sapiens | |||
2. | ALA520037 | 15e | INH | = | 8 | % | ALA5252730 | % | Homo sapiens | |||
3. | Neratinib (HKI-272) | 25o (table 3) | IC50 | = | 274 | nM | ALA5252710 | 6.56 | nM | Homo sapiens | ||
4. | ALA1090360 | 26 | IC50 | = | 310 | nM | ALA5252708 | 6.51 | nM | Homo sapiens | ||
5. | ALA3646210 | BDBM121388 | IC50 | = | 50 | nM | ALA5252708 | 7.30 | nM | Homo sapiens | ||
6. | ALA1997822 | SID103904321 | IC50 | = | 40 | nM | ALA5252708 | 7.40 | nM | Homo sapiens | ||
7. | ilorasertib | SID103904272 | IC50 | = | 13 | nM | ALA5252708 | 7.89 | nM | Homo sapiens | ||
8. | ALA5283398 | Fig 5, Cpd 2 | IC50 | = | 280 | nM | ALA5252708 | 6.55 | nM | Homo sapiens | ||
9. | ALA1807710 | 13 | INH | = | 66 | % | ALA5252698 | % | Homo sapiens | |||
10. | ALA1808262 | 24 | INH | = | 0.9 | % | ALA5252698 | % | Homo sapiens | |||
11. | Dabrafenib | 7, GSK2118436 | INH | = | 7 | % | ALA5252698 | % | Homo sapiens | |||
12. | ALA156218 | 6 | INH | = | 10 | % | ALA5252698 | % | Homo sapiens | |||
13. | ALA350702 | 6 | INH | = | 0 | % | ALA5252698 | % | Homo sapiens | |||
14. | ALA346551 | 6 | INH | = | 0 | % | ALA5252698 | % | Homo sapiens | |||
15. | ALA347419 | 6 | INH | = | 12 | % | ALA5252698 | % | Homo sapiens | |||
16. | ALA156506 | 6 | INH | = | 10 | % | ALA5252698 | % | Homo sapiens | |||
17. | ALA347857 | 6 | INH | = | 7 | % | ALA5252698 | % | Homo sapiens | |||
18. | ALA347632 | 6 | INH | = | 0 | % | ALA5252698 | % | Homo sapiens | |||
19. | ALA156684 | 6 | INH | = | 3 | % | ALA5252698 | % | Homo sapiens | |||
20. | ALA347647 | 6 | INH | = | 73 | % | ALA5252698 | % | Homo sapiens |