Activities

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Activities

Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA2425654	3	INH	=	87	%	ALA2429506			%	Homo sapiens
2.	ALA2425652	4	INH	<	50	%	ALA2429506			%	Homo sapiens
3.	ALA2425649	8	INH	=	78	%	ALA2429506			%	Homo sapiens
4.	ALA2425645	11	INH	=	88	%	ALA2429506			%	Homo sapiens
5.	ALA2425644	13	INH	=	96	%	ALA2429506			%	Homo sapiens
6.	ALA2425628	24f	Kd	=	0.87	uM	ALA2429181	6.06		nM	Homo sapiens
7.	ALA2425628	24f	INH	>	85	%	ALA2429506			%	Homo sapiens
8.	ALA2425646	12	INH	=	77	%	ALA2429506			%	Homo sapiens
9.	ALA2402081	37	INH	=	4	%	ALA2404336			%	Homo sapiens
10.	ALA2380845	17	IC50	=	36	nM	ALA2382839	7.44		nM	Homo sapiens
11.	ALA2380834	39	IC50	=	18	nM	ALA2382839	7.75		nM	Homo sapiens
12.	1-ethyl-3-[5-[6-(4-methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]urea	31	INH		0		ALA2071846		Dose-dependent effect	%	Homo sapiens
13.	N-[5-[6-(2,6-dichloro-4-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]acetamide	35	IC50	=	30	nM	ALA2071839	7.52		nM	Homo sapiens
14.	ALA2070618	34	IC50	=	32	nM	ALA2071839	7.50		nM	Homo sapiens
15.	ALA2070617	33	IC50	=	284	nM	ALA2071839	6.55		nM	Homo sapiens
16.	ALA2070616	32	IC50	=	87	nM	ALA2071839	7.06		nM	Homo sapiens
17.	1-ethyl-3-[5-[6-(4-methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]urea	31	IC50	=	58	nM	ALA2071839	7.24		nM	Homo sapiens
18.	ALA2070614	30	IC50	=	23	nM	ALA2071839	7.64		nM	Homo sapiens
19.	1-[5-[6-(2,6-dimethyl-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]-3-methylurea	29	IC50	=	66	nM	ALA2071839	7.18		nM	Homo sapiens
20.	ALA2070612	28	IC50	=	172	nM	ALA2071839	6.76		nM	Homo sapiens