Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Assay	Assay Organism
1.	ALA5270581	18	INH	>	50	nM	ALA5252873		nM	Homo sapiens
2.	ALA5278465	33	IC50	>	2	uM	ALA5252873		nM	Homo sapiens
3.	ALA5288565	29	IC50	>	2	uM	ALA5252873		nM	Homo sapiens
4.	Selitrectinib (LOXO-195)	SELITRECTINIB	% of control	=	10	%	ALA5213057		%	Homo sapiens
5.	Lorlatinib	8k, PF-06463922	Ki	=	17	nM	ALA5213164	7.77	nM	Homo sapiens
6.	XMD8-92	18	IC50	=	18	uM	ALA5213122	4.75	nM	Homo sapiens
7.	MPS1-IN-1	Mps1-IN-1	IC50	=	3100	nM	ALA5212773	5.51	nM	Homo sapiens
8.	ALA5175977	28	IC50	>	10	uM	ALA5165282		nM	Homo sapiens
9.	PF-543	PF-543	IC50	>	10	uM	ALA5165282		nM	Homo sapiens
10.	ALA5188399	1	Activity	<=	70	%	ALA5155256		%	Homo sapiens
11.	larotrectinib	LAROTRECTINIB	IC50	=	576	nmol/L	ALA5150441	6.24	nM	Homo sapiens
12.	ALA5170855	17b	Activity	=	0.1	%	ALA5129165		%	Homo sapiens
13.	ALA4458435	23; PF-06700841	INH	=	82	%	ALA4411556		%	Homo sapiens
14.	ALA4455923	48c	INH	<	50	%	ALA4405250		%	Homo sapiens
15.	BMS-690514	BMS-690514	Kd	<	225	nM	ALA4394545		nM	Homo sapiens
16.	ALA4559936	(+/-)-6	Activity	=	100	%	ALA4391617		%	Homo sapiens
17.	ALA4564973	50	INH	=	100	%	ALA4389991		%	Homo sapiens
18.	ALA4555459	43	INH	=	100	%	ALA4389514		%	Homo sapiens
19.	ALA4545456	24	INH	=	5	%	ALA4387369		%	Homo sapiens
20.	Abemaciclib	ABEMACICLIB	INH	=	2.4	%	ALA4387369		%	Homo sapiens