# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1233528 | VOLASERTIB | Kd | = | 195 | nM | ALA5213103 | 6.71 | nM | Homo sapiens | ||
2. | CC-671 | 23; CC-671 | IC50 | = | 1.1 | uM | ALA5213074 | 5.96 | nM | Homo sapiens | ||
3. | BI 2536 | 1 | % of control | = | 3.4 | % | ALA5213541 | % | Homo sapiens | |||
4. | ALA4745471 | EUB0000167b | IC50 | = | 30 | nM | ALA5210471 | 7.52 | nM | Homo sapiens | ||
5. | ALA4787282 | EUB0000168b | IC50 | > | 27000 | nM | ALA5210464 | nM | Homo sapiens | |||
6. | ALA4745471 | EUB0000167b | IC50 | = | 1600 | nM | ALA5210024 | 5.80 | nM | Homo sapiens | ||
7. | ALA4787282 | EUB0000168b | IC50 | > | 10000 | nM | ALA5210020 | nM | Homo sapiens | |||
8. | BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 1.5 | C | ALA5209700 | C | Homo sapiens | |||
9. | Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 1.84 | C | ALA5209700 | C | Homo sapiens | |||
10. | AZD6482 | AZD-6482 | Delta TM | = | 0.63 | C | ALA5209700 | C | Homo sapiens | |||
11. | ASP3026 | ASP-3026 | Delta TM | = | 8.23 | C | ALA5209700 | C | Homo sapiens | |||
12. | TC ASK 10 | EUB0000623aCl | Delta TM | = | 4.55 | C | ALA5209700 | C | Homo sapiens | |||
13. | AP26113 | AP26113 | Delta TM | = | 14.76 | C | ALA5209700 | C | Homo sapiens | |||
14. | AIM-100 | 2 | Delta TM | = | 2.62 | C | ALA5209700 | C | Homo sapiens | |||
15. | BMS-509744 | 3 | Delta TM | = | 7.16 | C | ALA5209700 | C | Homo sapiens | |||
16. | Selonsertib (GS-4997) | SELONSERTIB | Delta TM | = | 11.57 | C | ALA5209700 | C | Homo sapiens | |||
17. | SB590885 | 33, SB-590885 | Delta TM | = | 0.09 | C | ALA5209700 | C | Homo sapiens | |||
18. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | 2.73 | C | ALA5209700 | C | Homo sapiens | |||
19. | ALA3040440 | 1, 15 | Delta TM | = | 7.76 | C | ALA5209700 | C | Homo sapiens | |||
20. | NMS-P715 | 15, NMS-P715 | Delta TM | = | 4.44 | C | ALA5209700 | C | Homo sapiens |