# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TH 257 | EUB0000232b | Kd | > | 10 | uM | ALA5214768 | nM | Homo sapiens | |||
2. | TH 257 | EUB0000232b | % of control | = | 0 | % | ALA5214767 | % | Homo sapiens | |||
3. | GW843682X | 2 | % of control | = | 0.3 | % | ALA5213201 | % | Homo sapiens | |||
4. | BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | -0.42 | C | ALA5209780 | C | Homo sapiens | |||
5. | Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 1.19 | C | ALA5209780 | C | Homo sapiens | |||
6. | AZD6482 | AZD-6482 | Delta TM | = | 0.55 | C | ALA5209780 | C | Homo sapiens | |||
7. | ASP3026 | ASP-3026 | Delta TM | = | 3.07 | C | ALA5209780 | C | Homo sapiens | |||
8. | TC ASK 10 | EUB0000623aCl | Delta TM | = | -0.41 | C | ALA5209780 | C | Homo sapiens | |||
9. | AP26113 | AP26113 | Delta TM | = | 3.3 | C | ALA5209780 | C | Homo sapiens | |||
10. | AIM-100 | 2 | Delta TM | = | 3.82 | C | ALA5209780 | C | Homo sapiens | |||
11. | Selonsertib (GS-4997) | SELONSERTIB | Delta TM | = | -0.52 | C | ALA5209780 | C | Homo sapiens | |||
12. | SB590885 | 33, SB-590885 | Delta TM | = | 2.36 | C | ALA5209780 | C | Homo sapiens | |||
13. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | -1.29 | C | ALA5209780 | C | Homo sapiens | |||
14. | ALA3040440 | 1, 15 | Delta TM | = | -0.26 | C | ALA5209780 | C | Homo sapiens | |||
15. | NMS-P715 | 15, NMS-P715 | Delta TM | = | -1.96 | C | ALA5209780 | C | Homo sapiens | |||
16. | ALA4757879 | EUB0000633a | Delta TM | = | -1.14 | C | ALA5209780 | C | Homo sapiens | |||
17. | LDC 000067 | 5, LDC000067 | Delta TM | = | 0.4 | C | ALA5209780 | C | Homo sapiens | |||
18. | ALA4746004 | EUB0000617aCl | Delta TM | = | -1.15 | C | ALA5209780 | C | Homo sapiens | |||
19. | ALA1852688 | 5625 | Delta TM | = | 0.89 | C | ALA5209780 | C | Homo sapiens | |||
20. | HKI 357 | 7f (table 3) | Delta TM | = | 6.2 | C | ALA5209780 | C | Homo sapiens |