# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Canertinib (CI-1033) | 18 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
2. | Vandetanib | 22 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
3. | Erlotinib | Tarceva | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
4. | Gefitinib (ZD1839) | Iressa | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
5. | Imatinib (STI571) | 1 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
6. | ALA1725279 | SP-600125 | Kd | = | 0.22 | uM | ALA860649 | 6.66 | nM | Mus musculus | ||
7. | Doramapimod | 45 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
8. | VX-745 | 3 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
9. | SB 203580 (DMSO solution) | 9 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
10. | SB 202190 | 13 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
11. | Staurosporine | 1 (Staurosporine) | Kd | = | 0 | uM | ALA860649 | 9.82 | nM | Mus musculus | ||
12. | Flavopiridol | 1 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
13. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
14. | MnTMPyP pentachloride | 5 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
15. | ALA91829 | 1 | Kd | = | 0.09 | uM | ALA860649 | 7.05 | nM | Mus musculus | ||
16. | Tandutinib (MLN518) | 75 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
17. | Sunitinib | 12b | Kd | = | 0.16 | uM | ALA860649 | 6.80 | nM | Mus musculus | ||
18. | Vatalanib base | 1 | Kd | 0 | ALA860649 | Not Active | Mus musculus | |||||
19. | Pelitinib | EKB-569 | Kd | = | 1.1 | uM | ALA860649 | 5.96 | nM | Mus musculus | ||
20. | Lapatinib | GW-572016 | Kd | 0 | ALA860649 | Not Active | Mus musculus |