| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 18.682 | ALA5304852 | Homo sapiens | |||||
| 2. | ALA5306285 | EUB0002235 | delta Tm | = | 0.335 | ALA5304852 | Not Active | Homo sapiens | ||||
| 3. |  ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 18.682 | ALA5304748 | Homo sapiens | |||||
| 4. | ALA5308262 | EUB0002234 | delta Tm | = | 0.214 | ALA5304748 | Not Active | Homo sapiens | ||||
| 5. |  ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 18.684 | ALA5304582 | Homo sapiens | |||||
| 6. | ALA5308250 | EUB0002186 | delta Tm | = | -0.192 | ALA5304582 | Not Active | Homo sapiens | ||||
| 7. |  ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 18.684 | ALA5304483 | Homo sapiens | |||||
| 8. | ALA5306577 | EUB0002354 | delta Tm | = | -0.103 | ALA5304483 | Not Active | Homo sapiens | ||||
| 9. |  Staurosporine | 1 (Staurosporine) | Kd | = | 1 | nM | ALA5252317 | 9.00 | nM | Homo sapiens | ||
| 10. |  ALA5271697 | 8a | INH | = | 30 | % | ALA5252306 | % | Homo sapiens | |||
| 11. | ALA5271697 | 8a | deltaTm | = | 5.3 | degrees C | ALA5252296 | degrees C | Homo sapiens | |||
| 12. | ALA5271697 | 8a | deltaTm | = | 5.8 | degrees C | ALA5252296 | degrees C | Homo sapiens | |||
| 13. |  ALA4518706 | EUB0000702 | % of control | = | 2.3 | % | ALA5213311 | % | Homo sapiens | |||
| 14. |  Skepinone-L | 2, Skepinone-L | % of control | = | 37 | % | ALA5213507 | % | Homo sapiens | |||
| 15. |  GW843682X | 2 | % of control | = | 1 | % | ALA5213197 | % | Homo sapiens | |||
| 16. |  ALA4458078 | 16; SGCAAK1-1N | Kd | > | 10000 | nM | ALA5210463 | nM | Homo sapiens | |||
| 17. |  SGC AAK1 1 | 25; SGC-AAK1-1 | Ki | = | 17 | nM | ALA5210461 | 7.77 | nM | Homo sapiens | ||
| 18. | SGC AAK1 1 | 25; SGC-AAK1-1 | IC50 | = | 1500 | nM | ALA5210205 | 5.82 | nM | Homo sapiens | ||
| 19. |  BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 1.79 | C | ALA5209689 | C | Homo sapiens | |||
| 20. |  Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 2.07 | C | ALA5209689 | C | Homo sapiens |
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