# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA1952329 | Table 2, R1C3 | IC50 | = | 363 | nM | ALA5237490 | 6.44 | nM | Homo sapiens | ||
2. | Imidazopyridazin 1 | imidazo[1,2-b]pyridazine 1 | IC50 | = | 1.8 | uM | ALA5237490 | 5.75 | nM | Homo sapiens | ||
3. | ALA5179988 | 3 | Kd | = | 0.2 | uM | ALA5160045 | 6.70 | nM | Homo sapiens | ||
4. | ALA5189523 | 9 | Kd | = | 7.4 | uM | ALA5160045 | 5.13 | nM | Homo sapiens | ||
5. | ALA5183704 | 22 | INH | = | 0 | % | ALA5119695 | % | Homo sapiens | |||
6. | ALA3979678 | BDBM238766 | Kd | = | 1.7 | nM | ALA4478508 | 8.77 | nM | Homo sapiens | ||
7. | ALA3896195 | BDBM238707 | IC50 | = | 0.1 | nM | ALA4478465 | 10.00 | nM | Homo sapiens | ||
8. | ALA3927716 | BDBM238706 | IC50 | = | 0.3 | nM | ALA4478465 | 9.52 | nM | Homo sapiens | ||
9. | ALA4572195 | 25 | IC50 | = | 0.6 | nM | ALA4478465 | 9.22 | nM | Homo sapiens | ||
10. | ALA4589855 | 24 | IC50 | = | 1 | nM | ALA4478465 | 9.00 | nM | Homo sapiens | ||
11. | ALA4587256 | 23 | IC50 | = | 0.9 | nM | ALA4478465 | 9.05 | nM | Homo sapiens | ||
12. | ALA3950704 | BDBM238767 | IC50 | = | 0.4 | nM | ALA4478465 | 9.40 | nM | Homo sapiens | ||
13. | ALA4546373 | 21 | IC50 | = | 5.2 | nM | ALA4478465 | 8.28 | nM | Homo sapiens | ||
14. | ALA4559238 | 20 | IC50 | = | 4.9 | nM | ALA4478465 | 8.31 | nM | Homo sapiens | ||
15. | ALA4530924 | 19 | IC50 | = | 7.4 | nM | ALA4478465 | 8.13 | nM | Homo sapiens | ||
16. | ALA3902148 | BDBM238724 | IC50 | = | 0.1 | nM | ALA4478465 | 10.00 | nM | Homo sapiens | ||
17. | ALA3979678 | BDBM238766 | IC50 | = | 0.2 | nM | ALA4478465 | 9.70 | nM | Homo sapiens | ||
18. | ALA4522524 | 16 | IC50 | = | 2.1 | nM | ALA4478465 | 8.68 | nM | Homo sapiens | ||
19. | ALA3979182 | BDBM238637 | IC50 | = | 0.1 | nM | ALA4478465 | 10.00 | nM | Homo sapiens | ||
20. | ALA4527131 | 15 | IC50 | = | 2.5 | nM | ALA4478465 | 8.60 | nM | Homo sapiens |