# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NVP-BHG712 | NVP-BHG712 | IC50 | = | 263 | nM | ALA5212808 | 6.58 | nM | Homo sapiens | ||
2. | Afatinib dimaleate | AFATINIB DIMALEATE | Kd | = | 340 | nM | ALA5214833 | 6.47 | nM | Homo sapiens | ||
3. | ALA4526341 | EUB0000736 | % of control | = | 3 | % | ALA5213891 | % | Homo sapiens | |||
4. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405356 | % | Homo sapiens | |||
5. | ALA4559936 | (+/-)-6 | Activity | = | 97 | % | ALA4391318 | % | Homo sapiens | |||
6. | ALA4564973 | 50 | INH | = | 99 | % | ALA4389692 | % | Homo sapiens | |||
7. | ALA4555459 | 43 | INH | = | 51 | % | ALA4389215 | % | Homo sapiens | |||
8. | ALA4473365 | 7c | Activity | = | 49 | % | ALA4382496 | % | Homo sapiens | |||
9. | GSK2983559 active metabolite | 5 | INH | = | 70 | % | ALA4367362 | % | Homo sapiens | |||
10. | ALA4875968 | VIB-MDA-009 | INH | = | 19 | % | ALA4808075 | % | Homo sapiens | |||
11. | ALA4855209 | VIB-MDA-008 | INH | = | 69 | % | ALA4808075 | % | Homo sapiens | |||
12. | ALA4847460 | VIB-MDA-007 | INH | = | 58 | % | ALA4808075 | % | Homo sapiens | |||
13. | ALA4855979 | VIB-MDA-006 | INH | = | 62 | % | ALA4808075 | % | Homo sapiens | |||
14. | ALA4870763 | VIB-MDA-005 | INH | = | 67 | % | ALA4808075 | % | Homo sapiens | |||
15. | ALA4853006 | VIB-MDA-004 | INH | = | 27 | % | ALA4808075 | % | Homo sapiens | |||
16. | ALA4859179 | VIB-MDA-002 | INH | = | 69 | % | ALA4808075 | % | Homo sapiens | |||
17. | Dasatinib | 2, BMS-354825 | Activity | = | 25 | % | ALA4807828 | % | Homo sapiens | |||
18. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807828 | % | Homo sapiens | |||
19. | ALA4867844 | C7 | Activity | = | 25 | % | ALA4807828 | % | Homo sapiens | |||
20. | Dasatinib | 2, BMS-354825 | Activity | = | 50 | % | ALA4807596 | % | Homo sapiens |