# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | URMC-099 | 1, URMC-099 | INH | 0 | ALA2438985 | Active | % | Homo sapiens | ||||
2. | CEP-1347 | 2 | INH | 0 | ALA2438985 | Active | % | Homo sapiens | ||||
3. | ALA2425654 | 3 | INH | < | 50 | % | ALA2429298 | % | Homo sapiens | |||
4. | ALA2425652 | 4 | INH | = | 92 | % | ALA2429298 | % | Homo sapiens | |||
5. | ALA2425649 | 8 | INH | < | 50 | % | ALA2429298 | % | Homo sapiens | |||
6. | ALA2425645 | 11 | INH | = | 79 | % | ALA2429298 | % | Homo sapiens | |||
7. | ALA2425644 | 13 | INH | = | 99 | % | ALA2429298 | % | Homo sapiens | |||
8. | ALA2425646 | 12 | INH | < | 50 | % | ALA2429298 | % | Homo sapiens | |||
9. | ALA2312140 | 1 | IC50 | = | 65 | nM | ALA2320000 | 7.19 | nM | Homo sapiens | ||
10. | ALA2312141 | 2 | IC50 | = | 290 | nM | ALA2320000 | 6.54 | nM | Homo sapiens | ||
11. | ALA2312142 | 3 | IC50 | = | 6 | nM | ALA2320000 | 8.22 | nM | Homo sapiens | ||
12. | ALA2312143 | 4 | IC50 | = | 5 | nM | ALA2320000 | 8.30 | nM | Homo sapiens | ||
13. | 4-methoxy-3-[2-[3-methoxy-4-(4-methylpiperazin-1-yl)anilino]pyridin-4-yl]benzonitrile | 5 | IC50 | = | 3 | nM | ALA2320000 | 8.52 | nM | Homo sapiens | ||
14. | ALA2312145 | 6 | IC50 | = | 4 | nM | ALA2320000 | 8.40 | nM | Homo sapiens | ||
15. | ALA2312146 | 7 | IC50 | = | 55 | nM | ALA2320000 | 7.26 | nM | Homo sapiens | ||
16. | ALA2312147 | 8 | IC50 | = | 11 | nM | ALA2320000 | 7.96 | nM | Homo sapiens | ||
17. | ALA2312148 | 9 | IC50 | = | 8 | nM | ALA2320000 | 8.10 | nM | Homo sapiens | ||
18. | ALA2312149 | 10 | IC50 | > | 1000 | nM | ALA2320000 | nM | Homo sapiens | |||
19. | ALA2312150 | 11 | IC50 | = | 41 | nM | ALA2320000 | 7.39 | nM | Homo sapiens | ||
20. | ALA2312151 | 12 | IC50 | = | 118 | nM | ALA2320000 | 6.93 | nM | Homo sapiens |