# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ro-0505124 | Ro-0505124 | INH | < | 50 | % | ALA1959412 | % | Mus musculus | |||
2. | ALA2425652 | 4 | INH | < | 50 | % | ALA2428346 | % | Mus musculus | |||
3. | ALA2425649 | 8 | INH | < | 50 | % | ALA2428346 | % | Mus musculus | |||
4. | Canertinib (CI-1033) | 18 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
5. | Vandetanib | 22 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
6. | Erlotinib | Tarceva | Kd | = | 0.63 | uM | ALA860640 | 6.20 | nM | Mus musculus | ||
7. | Gefitinib (ZD1839) | Iressa | Kd | = | 1.4 | uM | ALA860640 | 5.85 | nM | Mus musculus | ||
8. | Imatinib (STI571) | 1 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
9. | ALA1725279 | SP-600125 | Kd | = | 0.68 | uM | ALA860640 | 6.17 | nM | Mus musculus | ||
10. | Doramapimod | 45 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
11. | VX-745 | 3 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
12. | SB 203580 (DMSO solution) | 9 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
13. | SB 202190 | 13 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
14. | Staurosporine | 1 (Staurosporine) | Kd | = | 0.003 | uM | ALA860640 | 8.52 | nM | Mus musculus | ||
15. | Flavopiridol | 1 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
16. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
17. | MnTMPyP pentachloride | 5 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
18. | ALA91829 | 1 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
19. | Tandutinib (MLN518) | 75 | Kd | 0 | ALA860640 | Not Active | Mus musculus | |||||
20. | Sunitinib | 12b | Kd | = | 0.11 | uM | ALA860640 | 6.96 | nM | Mus musculus |