# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BFH772 | 1 | IC50 | > | 0.5 | uM | ALA5252782 | nM | Homo sapiens | |||
2. | BAW2881(NVP-BAW2881) | 2 | IC50 | > | 0.5 | uM | ALA5252782 | nM | Homo sapiens | |||
3. | Alsterpaullone | 28d | IC50 | > | 100 | uM | ALA5227477 | nM | Homo sapiens | |||
4. | Kenpaullone | 28a | IC50 | > | 1000 | uM | ALA5227477 | nM | Homo sapiens | |||
5. | ALA1614712 | 1; NVP-AEW541 | IC50 | = | 2.3 | uM | ALA5224253 | 5.64 | nM | Homo sapiens | ||
6. | ALA1091644 | OSI-906 | IC50 | = | 75 | nM | ALA5224251 | 7.12 | nM | Homo sapiens | ||
7. | BMS-777607 | 10, BMS-777607 | IC50 | > | 2 | uM | ALA5212870 | nM | Homo sapiens | |||
8. | Afatinib dimaleate | AFATINIB DIMALEATE | IC50 | > | 10 | uM | ALA5214834 | nM | Homo sapiens | |||
9. | PF-04217903 | SID103905666 | IC50 | > | 10 | uM | ALA5212848 | nM | Homo sapiens | |||
10. | MPS1-IN-1 | Mps1-IN-1 | IC50 | = | 470 | nM | ALA5212785 | 6.33 | nM | Homo sapiens | ||
11. | MPS1-IN-1 | Mps1-IN-1 | % of control | = | 0.15 | % | ALA5212784 | % | Homo sapiens | |||
12. | ALA1091644 | OSI-906 | IC50 | = | 75 | nM | ALA5210319 | 7.12 | nM | Homo sapiens | ||
13. | ALA1091644 | OSI-906 | IC50 | = | 21 | nM | ALA5209907 | 7.68 | nM | Homo sapiens | ||
14. | ALA5175977 | 28 | IC50 | > | 10 | uM | ALA5165284 | nM | Homo sapiens | |||
15. | PF-543 | PF-543 | IC50 | > | 10 | uM | ALA5165284 | nM | Homo sapiens | |||
16. | ALA5182403 | 39 | INH | = | 4 | % | ALA5161374 | % | Homo sapiens | |||
17. | ALA5172009 | 38 | INH | = | 64 | % | ALA5161374 | % | Homo sapiens | |||
18. | ALA5202029 | 20 | INH | = | 57 | % | ALA5161374 | % | Homo sapiens | |||
19. | CH7057288 | CH7057288 | IC50 | > | 10000 | nM | ALA5119511 | nM | Homo sapiens | |||
20. | ALA5186340 | 1 | IC50 | > | 10000 | nM | ALA5119511 | nM | Homo sapiens |