# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Etomidate | Etomidate | EC50 | = | 2.3 | uM | ALA870388 | 5.64 | nM | Xenopus sp. | ||
2. | ALA385026 | BzBzl-etomidate | EC50 | = | 0.22 | uM | ALA870388 | 6.66 | nM | Xenopus sp. | ||
3. | ALA215734 | TDBzl-etomidate | EC50 | = | 0.7 | uM | ALA870388 | 6.16 | nM | Xenopus sp. | ||
4. | [³H]azietomidate | Azietomidate | EC50 | = | 2.2 | uM | ALA870388 | 5.66 | nM | Xenopus sp. | ||
5. | ALA58416 | 2c (Z) | Response | = | 135 | % | ALA824188 | % | Xenopus sp. | |||
6. | ALA58416 | 2c (Z) | Response | = | 300 | % | ALA824189 | % | Xenopus sp. | |||
7. | Nicotine | 2 | Response | = | 100 | % | ALA824188 | % | Xenopus sp. | |||
8. | Nicotine | 2 | Response | = | 100 | % | ALA824189 | % | Xenopus sp. | |||
9. | ALA291442 | 3a (E) | Response | = | 38 | % | ALA824188 | % | Xenopus sp. | |||
10. | ALA291442 | 3a (E) | Response | 0 | % | ALA824190 | Not Determined | Xenopus sp. | ||||
11. | 3-Methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole | 4a | Response | = | 40 | % | ALA824188 | % | Xenopus sp. | |||
12. | 3-Methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole | 4a | Response | = | 24 | % | ALA824189 | % | Xenopus sp. | |||
13. | ALA291780 | 2a (Z) | Response | = | 51 | % | ALA824188 | % | Xenopus sp. | |||
14. | ALA291780 | 2a (Z) | Response | = | 171 | % | ALA824189 | % | Xenopus sp. | |||
15. | ALA282030 | 6a | IC50 | = | 6 | nM | ALA823359 | 8.22 | nM | Xenopus sp. | ||
16. | ALA277711 | 7c | IC50 | = | 130 | nM | ALA823359 | 6.89 | nM | Xenopus sp. | ||
17. | ZK 200775 | NPQX | IC50 | = | 31 | nM | ALA823359 | 7.51 | nM | Xenopus sp. | ||
18. | ALA281393 | 7b | IC50 | = | 130 | nM | ALA823359 | 6.89 | nM | Xenopus sp. | ||
19. | ALA277281 | 4a | IC50 | = | 29 | nM | ALA823359 | 7.54 | nM | Xenopus sp. | ||
20. | Tezampanel | (-)-LY-293559 | IC50 | = | 233 | nM | ALA823359 | 6.63 | nM | Xenopus sp. |