# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 2-Nitrophenyl Phenyl Sulfone | 4a | EC50 | = | 3.4 | uM | ALA5244740 | 5.47 | nM | Human immunodeficiency virus | ||
2. | ALA358207 | 8f | EC50 | = | 15.08 | uM | ALA5244740 | 4.82 | nM | Human immunodeficiency virus | ||
3. | ALA5288408 | 47; R100155 | Activity | = | 80 | % | ALA5244645 | % | Human immunodeficiency virus | |||
4. | ALA5288408 | 47; R100155 | Activity | = | 70 | % | ALA5244644 | % | Human immunodeficiency virus | |||
5. | ALA5288408 | 47; R100155 | Activity | = | 50 | % | ALA5244643 | % | Human immunodeficiency virus | |||
6. | ALA5267740 | 15 | IC50 | = | 2.86 | uM | ALA5241743 | 5.54 | nM | Human immunodeficiency virus | ||
7. | ALA5273135 | 213 | EC50 | = | 1 | nM | ALA5241381 | 9.00 | nM | Human immunodeficiency virus | ||
8. | ALA2112593 | 57 | EC50 | = | 3.4 | uM | ALA5241379 | 5.47 | nM | Human immunodeficiency virus | ||
9. | ALA161076 | 65; L-ddA | EC50 | = | 8.2 | uM | ALA5241379 | 5.09 | nM | Human immunodeficiency virus | ||
10. | ALA5285337 | 64; L-d4A | EC50 | = | 0.38 | uM | ALA5241379 | 6.42 | nM | Human immunodeficiency virus | ||
11. | ALA5269335 | 16 | EC50 | = | 1 | nM | ALA5237341 | 9.00 | nM | Human immunodeficiency virus | ||
12. | ALA5289058 | 15 | EC50 | = | 1 | nM | ALA5237341 | 9.00 | nM | Human immunodeficiency virus | ||
13. | ALA1237000 | 5, MK-0536 | EC50 | = | 1 | nM | ALA5237341 | 9.00 | nM | Human immunodeficiency virus | ||
14. | Raltegravir (MK-0518) | 1, raltegravir | EC50 | = | 22 | nM | ALA5237341 | 7.66 | nM | Human immunodeficiency virus | ||
15. | ALA5269335 | 16 | EC50 | = | 1 | nM | ALA5237340 | 9.00 | nM | Human immunodeficiency virus | ||
16. | ALA5289058 | 15 | EC50 | = | 1 | nM | ALA5237340 | 9.00 | nM | Human immunodeficiency virus | ||
17. | ALA1237000 | 5, MK-0536 | EC50 | = | 2 | nM | ALA5237340 | 8.70 | nM | Human immunodeficiency virus | ||
18. | Raltegravir (MK-0518) | 1, raltegravir | EC50 | = | 13 | nM | ALA5237340 | 7.89 | nM | Human immunodeficiency virus | ||
19. | ALA5269335 | 16 | FC | = | 1 | ALA5237339 | Human immunodeficiency virus | |||||
20. | ALA5289058 | 15 | FC | = | 1.5 | ALA5237339 | Human immunodeficiency virus |