# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2151066 | 7b, diastereomeric mixture | IC50 | = | 0.033 | uM | ALA2153943 | 7.48 | nM | Homo sapiens | ||
2. | ALA2153705 | 9b | IC50 | = | 0.42 | uM | ALA2153943 | 6.38 | nM | Homo sapiens | ||
3. | ALA2153711 | 11b | IC50 | = | 0.032 | uM | ALA2153943 | 7.50 | nM | Homo sapiens | ||
4. | ALA2153710 | 10b | IC50 | = | 1.07 | uM | ALA2153943 | 5.97 | nM | Homo sapiens | ||
5. | ALA2153709 | 6b, diastereomeric mixture | IC50 | = | 0.033 | uM | ALA2153943 | 7.48 | nM | Homo sapiens | ||
6. | ALA2153707 | 2b | IC50 | = | 0.018 | uM | ALA2153943 | 7.75 | nM | Homo sapiens | ||
7. | ALA2153704 | 8b | IC50 | = | 0.8 | uM | ALA2153943 | 6.10 | nM | Homo sapiens | ||
8. | ALA2153712 | 12b | IC50 | > | 100 | uM | ALA2153943 | nM | Homo sapiens | |||
9. | [³H]methotrexate | 138 | Ki | <= | 0.004 | nM | ALA3130225 | nM | Homo sapiens | |||
10. | Trimethoprim | 139 | Ki | = | 19070 | nM | ALA3130225 | 4.72 | nM | Homo sapiens | ||
11. | Iclaprim | Iclaprim | Ki | = | 775 | nM | ALA3130225 | 6.11 | nM | Homo sapiens | ||
12. | ALA3128020 | 15 | Ki | = | 1607 | nM | ALA3130225 | 5.79 | nM | Homo sapiens | ||
13. | ALA3128021 | 16 | Ki | = | 93 | nM | ALA3130225 | 7.03 | nM | Homo sapiens | ||
14. | ALA3128022 | 17 | Ki | = | 1101 | nM | ALA3130225 | 5.96 | nM | Homo sapiens | ||
15. | ALA3128023 | 18 | Ki | = | 943 | nM | ALA3130225 | 6.03 | nM | Homo sapiens | ||
16. | ALA3128024 | 19 | Ki | = | 723 | nM | ALA3130225 | 6.14 | nM | Homo sapiens | ||
17. | ALA3128025 | 20 | Ki | = | 1026 | nM | ALA3130225 | 5.99 | nM | Homo sapiens | ||
18. | ALA3128026 | 21 | Ki | = | 663 | nM | ALA3130225 | 6.18 | nM | Homo sapiens | ||
19. | ALA3128027 | 22 | Ki | = | 2922 | nM | ALA3130225 | 5.53 | nM | Homo sapiens | ||
20. | ALA3127911 | 23 | Ki | > | 5000 | nM | ALA3130225 | nM | Homo sapiens |