# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2442124 | (R)-10b | IC50 | = | 0.58 | uM | ALA2446873 | 6.24 | nM | Mus musculus | ||
2. | ALA2442124 | (R)-10b | Activity | = | 69.6 | % | ALA2446871 | % | Mus musculus | |||
3. | ALA2403833 | 16b | IC50 | = | 1190 | nM | ALA2406364 | 5.92 | nM | Mus musculus | ||
4. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | IC50 | = | 1336 | nM | ALA2406364 | 5.87 | nM | Mus musculus | ||
5. | ALA2403838 | 17e | IC50 | = | 1420 | nM | ALA2406364 | 5.85 | nM | Mus musculus | ||
6. | ALA2403847 | 15d | IC50 | = | 2460 | nM | ALA2406364 | 5.61 | nM | Mus musculus | ||
7. | LDK378 | 6, LDK378 | IC50 | = | 2477 | nM | ALA2406364 | 5.61 | nM | Mus musculus | ||
8. | ALA2403848 | 15e | IC50 | = | 2517 | nM | ALA2406364 | 5.60 | nM | Mus musculus | ||
9. | ALA2403842 | 17i | IC50 | = | 2737 | nM | ALA2406364 | 5.56 | nM | Mus musculus | ||
10. | ALA2403846 | 15c | IC50 | = | 2884 | nM | ALA2406364 | 5.54 | nM | Mus musculus | ||
11. | ALA2403845 | 15a | IC50 | = | 3013 | nM | ALA2406364 | 5.52 | nM | Mus musculus | ||
12. | ALA2403844 | 7 | IC50 | = | 3395 | nM | ALA2406364 | 5.47 | nM | Mus musculus | ||
13. | Crizotinib (PF-02341066) | 14, PF-2341066 | IC50 | = | 3479 | nM | ALA2406364 | 5.46 | nM | Mus musculus | ||
14. | ALA2403831 | 20 | IC50 | = | 3800 | nM | ALA2406364 | 5.42 | nM | Mus musculus | ||
15. | ALA2403835 | 17b | IC50 | = | 3855 | nM | ALA2406364 | 5.41 | nM | Mus musculus | ||
16. | ALA2403849 | 16a | IC50 | = | 3997 | nM | ALA2406364 | 5.40 | nM | Mus musculus | ||
17. | ALA2403827 | 18b | IC50 | = | 4005 | nM | ALA2406364 | 5.40 | nM | Mus musculus | ||
18. | ALA2403843 | 18a | IC50 | = | 4077 | nM | ALA2406364 | 5.39 | nM | Mus musculus | ||
19. | ALA2403834 | 17a | IC50 | = | 4120 | nM | ALA2406364 | 5.38 | nM | Mus musculus | ||
20. | ALA2403836 | 17c | IC50 | = | 4336 | nM | ALA2406364 | 5.36 | nM | Mus musculus |