| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2152293 | 9 | TGI | 0 | ALA2155650 | Active | Homo sapiens | |||||
| 2. | ALA2152293 | 9 | TGI | 0 | ALA2155649 | Active | Homo sapiens | |||||
| 3. |  ALA2152295 | 11, demycarosyl-3D-beta-D-digitoxosylmithramycin SDK | GI50 | = | 32 | nM | ALA2157532 | nM | Homo sapiens | |||
| 4. | ALA2152293 | 9 | GI50 | = | 20 | nM | ALA2157532 | nM | Homo sapiens | |||
| 5. |  (2S,3S)-2-[(2S,4R,5R,6R)-4-[(2R,4R,5R,6R)-5-[(2R,4S,5R,6R)-4,5-dihydroxy-4,6-dimethyloxan-2-yl]oxy-4-hydroxy-6-methyloxan-2-yl]oxy-5-hydroxy-6-methyloxan-2-yl]oxy-3-[(1S,3S,4R)-3,4-dihydroxy-1-methoxy-2-oxopentyl]-6-[(2S,4R,5R,6R)-4-[(2R,4R,5S,6R)-4,5-dih | Mithramycin | GI50 | = | 63 | nM | ALA2157532 | nM | Homo sapiens | |||
| 6. | ALA2152293 | 9 | pGI50 | = | 7.67 | ALA2157532 | nM | Homo sapiens | ||||
| 7. | ALA2152295 | 11, demycarosyl-3D-beta-D-digitoxosylmithramycin SDK | pGI50 | = | 7.52 | ALA2157532 | nM | Homo sapiens | ||||
| 8. |  ALA2152294 | 10,demycarosylmithramycin SDK | pGI50 | = | 7.08 | ALA2157532 | nM | Homo sapiens | ||||
| 9. |  ALA2152292 | 2 | pGI50 | = | 7.31 | ALA2157532 | nM | Homo sapiens | ||||
| 10. | ALA2152294 | 10,demycarosylmithramycin SDK | GI50 | = | 0.3 | uM | ALA2157524 | nM | Homo sapiens | |||
| 11. | ALA2152295 | 11, demycarosyl-3D-beta-D-digitoxosylmithramycin SDK | GI50 | = | 0.3 | uM | ALA2157524 | nM | Homo sapiens | |||
| 12. | ALA2152293 | 9 | GI50 | = | 0.3 | uM | ALA2157524 | nM | Homo sapiens | |||
| 13. |  ALA3125578 | 4a | Activity | = | 109.26 | % | ALA3132203 | % | Homo sapiens | |||
| 14. |  ALA3125579 | 5a | Activity | = | 80.43 | % | ALA3132203 | % | Homo sapiens | |||
| 15. |  ALA3125580 | 6a | Activity | = | 26.33 | % | ALA3132203 | % | Homo sapiens | |||
| 16. | ALA3125580 | 6a | GI50 | = | 1.87 | uM | ALA3130634 | nM | Homo sapiens | |||
| 17. |  ALA3125581 | 7a | Activity | = | 94.18 | % | ALA3132203 | % | Homo sapiens | |||
| 18. |  ALA3125567 | 8a | Activity | = | 97.46 | % | ALA3132203 | % | Homo sapiens | |||
| 19. |  ALA3125569 | 6b | Activity | = | 105.96 | % | ALA3132203 | % | Homo sapiens | |||
| 20. |  ALA3122063 | 2a | Activity | = | 102.01 | % | ALA3122413 | % | Homo sapiens |
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