# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 2,6-Dimethyl-4-(3-methyl-1H-indazol-5-yl)-1,4-dihydropyridine-3,5-dicarbonitrile(BAY-474) | EUB0000293 | IC90 | 56 | nM | ALA4880563 | Active | nM | Homo sapiens | |||
2. | ALA5174958 | 18a | IC50 | = | 1.9 | uM | ALA5104347 | 5.72 | nM | Homo sapiens | ||
3. | D6808 | 14; D6808 | INH | 0 | ALA5100279 | Active | % | Homo sapiens | ||||
4. | D6808 | 14; D6808 | INH | 0 | ALA5100278 | Active | % | Homo sapiens | ||||
5. | ALA5172104 | 9y | Ratio IC50 | = | 2.6 | ALA5100225 | Homo sapiens | |||||
6. | ALA5190062 | 15 | IC50 | = | 163.3 | nM | ALA5100224 | 6.79 | nM | Homo sapiens | ||
7. | D6808 | 14; D6808 | IC50 | = | 0.7 | nM | ALA5100224 | 9.15 | nM | Homo sapiens | ||
8. | ALA5175023 | 13 | IC50 | = | 38.5 | nM | ALA5100224 | 7.42 | nM | Homo sapiens | ||
9. | ALA5176316 | 12 | IC50 | = | 10020 | nM | ALA5100224 | 5.00 | nM | Homo sapiens | ||
10. | ALA5195042 | 11 | IC50 | = | 3010 | nM | ALA5100224 | 5.52 | nM | Homo sapiens | ||
11. | ALA5205446 | 10 | IC50 | = | 446.6 | nM | ALA5100224 | 6.35 | nM | Homo sapiens | ||
12. | ALA5170241 | 9ym | IC50 | = | 186.6 | nM | ALA5100224 | 6.73 | nM | Homo sapiens | ||
13. | ALA5179628 | 9yl | IC50 | = | 45.9 | nM | ALA5100224 | 7.34 | nM | Homo sapiens | ||
14. | ALA5170338 | 9yk | IC50 | = | 115.1 | nM | ALA5100224 | 6.94 | nM | Homo sapiens | ||
15. | ALA5191797 | 9yj | IC50 | = | 9.8 | nM | ALA5100224 | 8.01 | nM | Homo sapiens | ||
16. | ALA5177753 | 9yi | IC50 | = | 20.1 | nM | ALA5100224 | 7.70 | nM | Homo sapiens | ||
17. | ALA5203752 | 9yh | IC50 | = | 106.2 | nM | ALA5100224 | 6.97 | nM | Homo sapiens | ||
18. | ALA5204053 | 9yg | IC50 | = | 428.3 | nM | ALA5100224 | 6.37 | nM | Homo sapiens | ||
19. | ALA5169499 | 9yf | IC50 | = | 375.2 | nM | ALA5100224 | 6.43 | nM | Homo sapiens | ||
20. | ALA5185647 | 9ye | IC50 | = | 211.5 | nM | ALA5100224 | 6.67 | nM | Homo sapiens |