# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Clofarabine | Table I Row 6 | IC50 | = | 0.23 | uM | ALA5247117 | 6.64 | nM | Mus musculus | ||
2. | Fludarabine phosphate | Fludarabine Phosphate | IC50 | = | 3 | uM | ALA5247117 | 5.52 | nM | Mus musculus | ||
3. | Cladribine | 25 | IC50 | = | 0.07 | uM | ALA5247117 | 7.16 | nM | Mus musculus | ||
4. | ALA5269069 | 72 | IC50 | = | 2.6 | ug ml-1 | ALA5246037 | ug.mL-1 | Mus musculus | |||
5. | ALA5273132 | 70 | IC50 | = | 2.6 | ug ml-1 | ALA5246037 | ug.mL-1 | Mus musculus | |||
6. | ALA5274197 | 71 | IC50 | = | 2.6 | ug ml-1 | ALA5246037 | ug.mL-1 | Mus musculus | |||
7. | ALA5271541 | 18 | IC50 | = | 2.9 | uM | ALA5245838 | 5.54 | nM | Mus musculus | ||
8. | ALA5274310 | 17 | IC50 | = | 2.9 | uM | ALA5245838 | 5.54 | nM | Mus musculus | ||
9. | ALA5284911 | 80 | IC50 | = | 9 | nM | ALA5245838 | 8.05 | nM | Mus musculus | ||
10. | ALA5267070 | 27 | IC50 | = | 321 | uM | ALA5245838 | nM | Mus musculus | |||
11. | ALA5284753 | 26 | IC50 | = | 98 | uM | ALA5245838 | 4.01 | nM | Mus musculus | ||
12. | ALA5172923 | 3 | IC50 | = | 8.1 | uM | ALA5245838 | 5.09 | nM | Mus musculus | ||
13. | ALA5288713 | 24 | IC50 | = | 20.4 | uM | ALA5245838 | 4.69 | nM | Mus musculus | ||
14. | ALA5267470 | 16 | IC50 | = | 2.9 | uM | ALA5245838 | 5.54 | nM | Mus musculus | ||
15. | ALA5281013 | 10 | IC50 | = | 4.6 | ug ml-1 | ALA5245838 | ug.mL-1 | Mus musculus | |||
16. | ALA5278753 | 9 | INH | = | 90 | % | ALA5245837 | % | Mus musculus | |||
17. | ALA5284273 | 8 | INH | = | 70 | % | ALA5245837 | % | Mus musculus | |||
18. | ALA5284062 | 7 | INH | = | 40 | % | ALA5245837 | % | Mus musculus | |||
19. | ALA2148106 | DAT | INH | = | 50 | % | ALA5245837 | % | Mus musculus | |||
20. | ALA5267707 | 5 | INH | = | 25 | % | ALA5245837 | % | Mus musculus |