# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PD173074 | 12 | Activity | = | 1.04 | ALA975127 | Homo sapiens | |||||
2. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 1.005 | ALA975127 | Homo sapiens | |||||
3. | Imatinib (STI571) | 1 | Activity | = | 1.035 | ALA975127 | Homo sapiens | |||||
4. | Tozasertib | VX-680 | Activity | = | 0.96 | ALA975127 | Homo sapiens | |||||
5. | Neratinib (HKI-272) | 25o (table 3) | Activity | = | 0.874 | ALA975127 | Homo sapiens | |||||
6. | MnTMPyP pentachloride | 5 | Activity | = | 1.032 | ALA975127 | Homo sapiens | |||||
7. | PHA-665752 | PHA-665752 | Activity | = | 1.063 | ALA975127 | Homo sapiens | |||||
8. | Sunitinib | 12b | Activity | = | 0.858 | ALA975127 | Homo sapiens | |||||
9. | Erlotinib | Tarceva | Activity | = | 1.136 | ALA975127 | Homo sapiens | |||||
10. | Saracatinib (AZD0530) | 33, AZD-0530 | Activity | = | 0.848 | ALA975127 | Homo sapiens | |||||
11. | Crizotinib | 14, PF-2341066 | Activity | = | 1.048 | ALA975127 | Homo sapiens | |||||
12. | ALA148624 | II | IC50 | = | 4 | uM | ALA753975 | 5.40 | nM | Homo sapiens | ||
13. | ALA148624 | II | IC50 | = | 5.1 | uM | ALA857701 | 5.29 | nM | Homo sapiens | ||
14. | ALA148624 | II | IC50 | = | 6 | uM | ALA753974 | 5.22 | nM | Homo sapiens | ||
15. | ALA148734 | I | IC50 | = | 4.5 | uM | ALA753975 | 5.35 | nM | Homo sapiens | ||
16. | ALA148734 | I | IC50 | = | 6 | uM | ALA857701 | 5.22 | nM | Homo sapiens | ||
17. | ALA148734 | I | IC50 | = | 6.5 | uM | ALA753974 | 5.19 | nM | Homo sapiens | ||
18. | ALA148624 | II | IC50 | = | 14 | uM | ALA753975 | 4.85 | nM | Homo sapiens | ||
19. | ALA148624 | II | IC50 | = | 16 | uM | ALA857701 | 4.80 | nM | Homo sapiens | ||
20. | ALA148624 | II | IC50 | = | 18 | uM | ALA753974 | 4.75 | nM | Homo sapiens |