| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2148108 | 5, 10-methyl-aplog-1 | Activity | < | 10 | % | ALA2148235 | % | Homo sapiens | |||
| 2. |  ALA2148107 | 4, 4-methyl-aplog-1 | Activity | < | 10 | % | ALA2148235 | % | Homo sapiens | |||
| 3. |  ALA1258348 | 1 | Activity | 0 | ALA2148234 | Toxic | Homo sapiens | |||||
| 4. |  Phorbol 12-myristate 13-acetate | 1 | Activity | 0 | ALA2148235 | Toxic | Homo sapiens | |||||
| 5. |  ALA2148106 | DAT | Activity | 0 | ALA2148235 | Toxic | Homo sapiens | |||||
| 6. |  ALA1096256 | 1 | IC50 | = | 0.14 | uM | ALA3136327 | 6.85 | nM | Homo sapiens | ||
| 7. |  ALA3133719 | 2, DeAMDeBAA | IC50 | > | 10 | uM | ALA3136327 | nM | Homo sapiens | |||
| 8. |  ALA3133720 | 3, DeBUAA | IC50 | > | 10 | uM | ALA3136327 | nM | Homo sapiens | |||
| 9. |  ALA3133721 | 5, DeBAA, Debromoagelastatin A | IC50 | = | 3.16 | uM | ALA3136327 | 5.50 | nM | Homo sapiens | ||
| 10. |  ALA3133722 | 6, DeBEAA, Debromoethylagelastatin A | IC50 | 0 | ALA3136327 | Not Determined | Homo sapiens | |||||
| 11. |  ALA3133723 | 7, CAA, Chloroagelasttain A | IC50 | = | 0.18 | uM | ALA3136327 | 6.75 | nM | Homo sapiens | ||
| 12. |  ALA3133724 | 8, CEAA, Chloroethylagelastatin A | IC50 | = | 0.3 | uM | ALA3136327 | 6.52 | nM | Homo sapiens | ||
| 13. |  ALA3133725 | 9, DCEAA, Dichloroethylagelastatin A | IC50 | = | 0.62 | uM | ALA3136327 | 6.21 | nM | Homo sapiens | ||
| 14. |  ALA3133726 | 10, EAA, Ethylagelastatin A | IC50 | 0 | ALA3136327 | Not Determined | Homo sapiens | |||||
| 15. |  ALA3133727 | 14, N-PMBAA, N-p-methoxybenzylagelasttain A | IC50 | 0 | ALA3136327 | Not Determined | Homo sapiens | |||||
| 16. |  ALA3133728 | 15, CPAA, Cyclopropylagelastatin | IC50 | = | 0.4 | uM | ALA3136327 | 6.40 | nM | Homo sapiens | ||
| 17. |  ALA3133729 | 16, PAA, Phenylagelastatin A | IC50 | = | 3.8 | uM | ALA3136327 | 5.42 | nM | Homo sapiens | ||
| 18. |  ALA3133730 | 17, APAA, Aminophenylagelastatin A | IC50 | 0 | ALA3136327 | Not Determined | Homo sapiens | |||||
| 19. |  ALA3133717 | 18, UAA, Urea agelastatin A | IC50 | > | 10 | uM | ALA3136327 | nM | Homo sapiens | |||
| 20. |  ALA3133718 | 19, ent-AA | IC50 | 0 | ALA3136327 | Not Determined | Homo sapiens |
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