# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2430263 | 21 | IC50 | = | 3.56 | uM | ALA2434175 | 5.45 | nM | Homo sapiens | ||
2. | tafetinib | 61, SIM010603 | IC50 | = | 3.31 | uM | ALA2434175 | 5.48 | nM | Homo sapiens | ||
3. | ALA2430264 | 23 | IC50 | = | 1.83 | uM | ALA2434175 | 5.74 | nM | Homo sapiens | ||
4. | ALA2430266 | 25 | IC50 | 0 | ALA2434175 | Not Determined | Homo sapiens | |||||
5. | Sunitinib | 12b | IC50 | = | 2.44 | uM | ALA2434175 | 5.61 | nM | Homo sapiens | ||
6. | ALA2385603 | 3 | IC50 | = | 0.016 | uM | ALA2388618 | 7.80 | nM | Homo sapiens | ||
7. | ALA2385602 | 2 | IC50 | = | 0.042 | uM | ALA2388618 | 7.38 | nM | Homo sapiens | ||
8. | ALA2385603 | 3 | IC50 | > | 10 | uM | ALA2388617 | nM | Homo sapiens | |||
9. | ALA2385602 | 2 | IC50 | > | 10 | uM | ALA2388617 | nM | Homo sapiens | |||
10. | ALA2385602 | 2 | Ratio IC50 | = | 240 | ALA2388616 | Homo sapiens | |||||
11. | ALA2385603 | 3 | Ratio IC50 | = | 240 | ALA2388616 | Homo sapiens | |||||
12. | ALA72974 | 8c | IC50 | = | 0.17 | nM | ALA2379120 | 9.77 | nM | Homo sapiens | ||
13. | ALA419083 | 8e | IC50 | = | 0.32 | nM | ALA2379120 | 9.49 | nM | Homo sapiens | ||
14. | Diflomotecan | 8f | IC50 | = | 0.4 | nM | ALA2379120 | 9.40 | nM | Homo sapiens | ||
15. | ALA306721 | 8a | IC50 | = | 1.6 | nM | ALA2379120 | 8.80 | nM | Homo sapiens | ||
16. | ALA74190 | hCPT | IC50 | = | 3.3 | nM | ALA2379120 | 8.48 | nM | Homo sapiens | ||
17. | ALA306796 | 8b | IC50 | = | 4.5 | nM | ALA2379120 | 8.35 | nM | Homo sapiens | ||
18. | ALA74863 | 8d | IC50 | = | 22 | nM | ALA2379120 | 7.66 | nM | Homo sapiens | ||
19. | ALA2377447 | 12-Cl-hCPT | FC | = | 23 | ALA2379119 | Homo sapiens | |||||
20. | (S)-(+)-Camptothecin | Camptothecin | IC50 | = | 88 | nM | ALA2379120 | 7.06 | nM | Homo sapiens |