# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 5-Fluorouracil | FUra | TGI | = | 41 | % | ALA3280698 | % | Rattus norvegicus | |||
2. | FT-207 (NSC 148958) | 2 | TGI | = | 52 | % | ALA3280697 | % | Rattus norvegicus | |||
3. | ALA3272516 | 4, Thf2-FU | TGI | = | 58 | % | ALA3280697 | % | Rattus norvegicus | |||
4. | FT-207 (NSC 148958) | 2 | TGI | = | 32 | % | ALA3280355 | % | Rattus norvegicus | |||
5. | ALA3272516 | 4, Thf2-FU | TGI | = | 43 | % | ALA3280355 | % | Rattus norvegicus | |||
6. | ALA3272485 | (S)-(-)-Thf-FU | TGI | = | 40.6 | % | ALA3279676 | % | Rattus norvegicus | |||
7. | FT-207 (NSC 148958) | 2 | TGI | = | 38.9 | % | ALA3279676 | % | Rattus norvegicus | |||
8. | ALA235993 | SID430704 | TGI | = | 33.7 | % | ALA3279676 | % | Rattus norvegicus | |||
9. | ALA235993 | SID430704 | Activity | = | 2.42 | g | ALA3279675 | g | Rattus norvegicus | |||
10. | FT-207 (NSC 148958) | 2 | Activity | = | 2.23 | g | ALA3279675 | g | Rattus norvegicus | |||
11. | ALA3272485 | (S)-(-)-Thf-FU | Activity | = | 2.17 | g | ALA3279675 | g | Rattus norvegicus | |||
12. | ALA79188 | 1 | Inhibition | = | 94 | % | ALA821054 | % | Rattus norvegicus | |||
13. | ALA322225 | 4 | IC50 | = | 660 | nM | ALA821051 | 6.18 | nM | Rattus norvegicus | ||
14. | GMX1778 | CHS 828 | IC50 | = | 140 | nM | ALA821051 | 6.85 | nM | Rattus norvegicus | ||
15. | Paclitaxel | Paclitaxel | IC50 | = | 7.9 | nM | ALA821051 | 8.10 | nM | Rattus norvegicus | ||
16. | Daunorubicin-¹³C,d3 | Daunorubicin | IC50 | = | 7.4 | nM | ALA821051 | 8.13 | nM | Rattus norvegicus |