# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | digoxin | Digoxin | IC50 | = | 10 | nM | ALA5097072 | 8.00 | nM | Homo sapiens | ||
2. | AEE788 (NVP-AEE788) | GNF-Pf-5343 | IC50 | = | 3.8 | uM | ALA5097068 | 5.42 | nM | Homo sapiens | ||
3. | Tolfenamic Acid | Tolfenamic acid | IC50 | = | 20.8 | ug ml-1 | ALA5097066 | ug.mL-1 | Homo sapiens | |||
4. | ALA406658 | 18 | IC50 | = | 4.89 | uM | ALA5097065 | 5.31 | nM | Homo sapiens | ||
5. | BKM120 | 15, NVP-BKM120 | IC50 | = | 0.279 | uM | ALA5097042 | 6.55 | nM | Homo sapiens | ||
6. | ALA2105763 | QUISINOSTAT | IC50 | < | 200 | nM | ALA5097031 | nM | Homo sapiens | |||
7. | LAQ824 | 9 | IC50 | < | 200 | nM | ALA5097031 | nM | Homo sapiens | |||
8. | ALA5187942 | 5 | Activity | 0 | ALA5164305 | Active | Homo sapiens | |||||
9. | ALA5187942 | 5 | Activity | 0 | ALA5164304 | Active | Homo sapiens | |||||
10. | Rucaparib | 63, AG-014699 | IC50 | = | 62.065 | uM | ALA2363167 | 4.21 | nM | Homo sapiens | ||
11. | CCT 018159 | 3a CCT018159 | IC50 | = | 16.399 | uM | ALA2363167 | 4.79 | nM | Homo sapiens | ||
12. | TW-37 | 5, TW-37 | IC50 | = | 0.284 | uM | ALA2363167 | 6.55 | nM | Homo sapiens | ||
13. | JNJ-26854165 (Serdemetan) | SID137276015 | IC50 | = | 12.61 | uM | ALA2363167 | 4.90 | nM | Homo sapiens | ||
14. | PF-4708671 | SID137275978 | IC50 | = | 490.239 | uM | ALA2363167 | nM | Homo sapiens | |||
15. | Avagacestat | 80 BMS-708163 | IC50 | = | 53.344 | uM | ALA2363167 | 4.27 | nM | Homo sapiens | ||
16. | EHT 1864 | SID137275837 | IC50 | = | 361.934 | uM | ALA2363167 | nM | Homo sapiens | |||
17. | CCT007093 | A17 | IC50 | = | 266.577 | uM | ALA2363167 | nM | Homo sapiens | |||
18. | AZD6482 | AZD-6482 | IC50 | = | 33.497 | uM | ALA2363167 | 4.47 | nM | Homo sapiens | ||
19. | ALA1614701 | AZD-6244 | IC50 | = | 79.819 | uM | ALA2363167 | 4.10 | nM | Homo sapiens | ||
20. | SB590885 | 33, SB-590885 | IC50 | = | 46.09 | uM | ALA2363167 | 4.34 | nM | Homo sapiens |