# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4642465 | 1 | GI50 | = | 0.02 | uM | ALA4614889 | nM | Homo sapiens | |||
2. | Matrine | 2 | Activity | = | 56.1 | % | ALA4327205 | % | Homo sapiens | |||
3. | Matrine | 2 | GI | = | 47.2 | % | ALA4327204 | % | Homo sapiens | |||
4. | Matrine | 2 | GI | = | 38 | % | ALA4327203 | % | Homo sapiens | |||
5. | Matrine | 2 | GI | = | 59.3 | % | ALA4327202 | % | Homo sapiens | |||
6. | Matrine | 2 | GI | = | 47.5 | % | ALA4327201 | % | Homo sapiens | |||
7. | Matrine | 2 | GI | = | 28.3 | % | ALA4327200 | % | Homo sapiens | |||
8. | Matrine | 2 | GI | = | 12.7 | % | ALA4327199 | % | Homo sapiens | |||
9. | ALA49378 | PBR-MEL | GSH | = | 33.2 | uM g-1 | ALA664746 | uM g-1 | Homo sapiens | |||
10. | ALA49378 | PBR-MEL | GSH | = | 17.5 | uM g-1 | ALA663794 | uM g-1 | Homo sapiens | |||
11. | ALA49378 | PBR-MEL | GST activity | = | 327.9 | nM min-1 (mg of protein)-1 | ALA664747 | nM min-1 (mg of protein)-1 | Homo sapiens | |||
12. | ALA49378 | PBR-MEL | GST activity | = | 212.6 | nM min-1 (mg of protein)-1 | ALA663795 | nM min-1 (mg of protein)-1 | Homo sapiens | |||
13. | ALA49378 | PBR-MEL | IC50 | = | 32.8 | uM | ALA663793 | 4.48 | nM | Homo sapiens | ||
14. | ALA49378 | PBR-MEL | IC50 | = | 25 | uM | ALA663796 | 4.60 | nM | Homo sapiens | ||
15. | ALA523 | 3 | IC50 | > | 200 | uM | ALA663793 | nM | Homo sapiens | |||
16. | ALA523 | 3 | IC50 | > | 200 | uM | ALA663796 | nM | Homo sapiens | |||
17. | Melphalan | melphalan | IC50 | = | 52.4 | uM | ALA663793 | 4.28 | nM | Homo sapiens | ||
18. | Melphalan | melphalan | IC50 | = | 12.4 | uM | ALA663796 | 4.91 | nM | Homo sapiens |