# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PACMA 31 | P; PACMA31 | INH | 0 | ALA4390891 | Not Active | % | Homo sapiens | ||||
2. | ALA4464788 | 68 | INH | 0 | ALA4390890 | Active | % | Homo sapiens | ||||
3. | ALA4545330 | 6; BAP2 | INH | 0 | ALA4390890 | Active | % | Homo sapiens | ||||
4. | ALA5187858 | 1a | Activity | = | 15 | % | ALA5121785 | % | Homo sapiens | |||
5. | ALA5089694 | 6s | IC50 | = | 9.9 | uM | ALA5046928 | 5.00 | nM | Homo sapiens | ||
6. | ALA5084156 | 6r | IC50 | = | 17.3 | uM | ALA5046928 | 4.76 | nM | Homo sapiens | ||
7. | [³H]methotrexate | 138 | IC50 | = | 16 | nM | ALA663147 | 7.80 | nM | Homo sapiens | ||
8. | trimetrexate | TMQ | IC50 | = | 60 | nM | ALA663147 | 7.22 | nM | Homo sapiens | ||
9. | piritrexim | 6 | IC50 | = | 230 | nM | ALA663147 | 6.64 | nM | Homo sapiens | ||
10. | ALA170758 | 5o | IC50 | = | 4.6 | nM | ALA663147 | 8.34 | nM | Homo sapiens |