# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5208121 | 12 | Activity | = | 21.5 | % | ALA5151564 | % | Homo sapiens | |||
2. | ALA5170058 | 11 | Activity | = | 16.7 | % | ALA5151564 | % | Homo sapiens | |||
3. | ALA5198503 | 10 | Activity | = | 17.4 | % | ALA5151564 | % | Homo sapiens | |||
4. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | IC50 | > | 2 | uM | ALA4415374 | nM | Homo sapiens | |||
5. | N-(4-{3-[2-(methylcarbamoyl)ethyl]-5-[4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl]-1H-pyrazol-1-yl}phenyl)prop-2-ynamide | 1; Tr-87 | IC50 | > | 2 | uM | ALA4415368 | nM | Homo sapiens | |||
6. | ALA4468410 | 18 | GI | = | 45.5 | % | ALA4386867 | % | Homo sapiens | |||
7. | ALA4468410 | 18 | GI | = | 53.8 | % | ALA4386866 | % | Homo sapiens | |||
8. | ALA4468410 | 18 | GI | = | 57.3 | % | ALA4386865 | % | Homo sapiens | |||
9. | ALA4468410 | 18 | GI | = | 65 | % | ALA4386864 | % | Homo sapiens | |||
10. | Vincristine | Vincristine | IC50 | = | 1.03 | uM | ALA4375930 | 5.99 | nM | Homo sapiens | ||
11. | ALA4464038 | 87a | IC50 | = | 1.73 | uM | ALA4375930 | 5.76 | nM | Homo sapiens | ||
12. | ALA4452542 | 87-9 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
13. | ALA4473974 | 87-8 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
14. | ALA4459992 | 87-7 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
15. | ALA4519233 | 87-6 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
16. | ALA4563218 | 87-5 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
17. | ALA4434896 | 87-4 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
18. | ALA4539544 | 87-3 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
19. | ALA4441645 | 87-2 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens | ||
20. | ALA4439249 | 87-1 | IC50 | = | 1.01 | uM | ALA4375930 | 6.00 | nM | Homo sapiens |