# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA25889 | DMPDDF | Uptake | = | 85 | % | ALA688846 | % | Rattus norvegicus | |||
2. | ALA25889 | DMPDDF | Uptake | = | 100 | % | ALA688844 | % | Rattus norvegicus | |||
3. | ALA25889 | DMPDDF | Uptake | = | 25 | % | ALA688986 | % | Rattus norvegicus | |||
4. | ALA25889 | DMPDDF | Uptake | = | 25 | % | ALA688847 | % | Rattus norvegicus | |||
5. | ALA25889 | DMPDDF | Uptake | = | 25 | % | ALA688987 | % | Rattus norvegicus | |||
6. | ALA25889 | DMPDDF | Uptake | = | 25 | % | ALA688845 | % | Rattus norvegicus | |||
7. | ALA25889 | DMPDDF | Uptake | = | 100 | % | ALA689456 | % | Rattus norvegicus | |||
8. | ALA25889 | DMPDDF | Uptake | = | 83 | % | ALA688984 | % | Rattus norvegicus | |||
9. | ALA25889 | DMPDDF | Uptake | = | 90 | % | ALA688982 | % | Rattus norvegicus | |||
10. | ALA25889 | DMPDDF | Uptake | = | 22 | % | ALA690437 | % | Rattus norvegicus | |||
11. | ALA25889 | DMPDDF | Uptake | = | 22 | % | ALA688985 | % | Rattus norvegicus | |||
12. | ALA25889 | DMPDDF | Uptake | = | 8.5 | % | ALA690438 | % | Rattus norvegicus | |||
13. | ALA25889 | DMPDDF | Uptake | = | 11 | % | ALA688983 | % | Rattus norvegicus | |||
14. | ALA25889 | DMPDDF | Uptake | = | 100 | % | ALA690544 | % | Rattus norvegicus | |||
15. | ALA25889 | DMPDDF | IC50 | = | 2240 | nM | ALA688483 | 5.65 | nM | Rattus norvegicus | ||
16. | Methotrexate | 138 | IC50 | = | 906 | nM | ALA688483 | 6.04 | nM | Rattus norvegicus | ||
17. | ALA422395 | 1a | IC50 | = | 2000 | nM | ALA688483 | 5.70 | nM | Rattus norvegicus | ||
18. | ALA344876 | 2 | Relative activity | = | 0.19 | ALA688481 | Rattus norvegicus | |||||
19. | ALA344876 | 2 | IC50 | = | 9.5 | uM | ALA688480 | 5.02 | nM | Rattus norvegicus | ||
20. | ALA3143620 | 3 | Relative activity | = | 0.15 | ALA688482 | Rattus norvegicus |