# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | GMX1778 | CHS 828 | IC50 | = | 2067 | nM | ALA5243297 | 5.68 | nM | Homo sapiens | ||
2. | ALA5267417 | 133a | IC50 | = | 282 | nM | ALA5243297 | 6.55 | nM | Homo sapiens | ||
3. | ALA5285409 | 24 | Activity | = | 55 | % | ALA5236995 | % | Homo sapiens | |||
4. | ALA5285409 | 24 | Activity | = | 38 | % | ALA5236994 | % | Homo sapiens | |||
5. | ALA5285409 | 24 | Activity | = | 60 | % | ALA5236993 | % | Homo sapiens | |||
6. | ALA5285409 | 24 | Activity | = | 41 | % | ALA5236992 | % | Homo sapiens | |||
7. | ALA5285409 | 24 | IC50 | = | 15.9 | uM | ALA5236991 | 4.80 | nM | Homo sapiens | ||
8. | ALA5285742 | 22 | IC50 | = | 0.41 | uM | ALA5236988 | 6.39 | nM | Homo sapiens | ||
9. | ALA4467135 | Apicidin | IC50 | = | 0.19 | uM | ALA4422823 | 6.72 | nM | Homo sapiens | ||
10. | TD52 | TD52 | INH | 0 | ALA4420539 | Not Active | % | Homo sapiens | ||||
11. | TD52 | TD52 | INH | 0 | ALA4420538 | Not Active | % | Homo sapiens | ||||
12. | TD52 | TD52 | INH | 0 | ALA4420537 | Not Active | % | Homo sapiens | ||||
13. | TD52 | TD52 | INH | 0 | ALA4420523 | Tde | % | Homo sapiens | ||||
14. | TD52 | TD52 | INH | 0 | ALA4420517 | Dose-dependent effect | % | Homo sapiens | ||||
15. | TD52 | TD52 | Ratio | = | 0.01 | ALA4420501 | Homo sapiens | |||||
16. | TD52 | TD52 | Ratio | = | 0.36 | ALA4420500 | Homo sapiens | |||||
17. | TD52 | TD52 | Ratio | = | 0.84 | ALA4420499 | Homo sapiens | |||||
18. | TD52 | TD52 | Ratio | = | 0.99 | ALA4420498 | Homo sapiens | |||||
19. | TD52 | TD52 | Activity | 0 | ALA4420461 | Active | Homo sapiens | |||||
20. | TD52 | TD52 | Activity | 0 | ALA4420486 | Dose-dependent effect | Homo sapiens |