# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SAR407899 | 14C | IC50 | = | 122 | nM | ALA5236742 | 6.91 | nM | Homo sapiens | ||
2. | FASUDIL | HA-1077 | IC50 | = | 1.3 | uM | ALA5236742 | 5.89 | nM | Homo sapiens | ||
3. | ALA4205860 | 23 | Activity | 0 | ALA4188461 | Not Active | Homo sapiens | |||||
4. | ALA4204145 | 24 | Activity | 0 | ALA4188461 | Not Active | Homo sapiens | |||||
5. | ALA4208156 | 25 | Activity | 0 | ALA4188461 | Not Active | Homo sapiens | |||||
6. | ALA4205860 | 23 | Activity | = | 92 | % | ALA4188462 | % | Homo sapiens | |||
7. | ALA4204145 | 24 | Activity | = | 100 | % | ALA4188462 | % | Homo sapiens | |||
8. | ALA4208156 | 25 | Activity | = | 97 | % | ALA4188463 | % | Homo sapiens | |||
9. | ALA2349065 | 1 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
10. | ALA2349064 | 2 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
11. | ALA2349063 | 3 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
12. | ALA2349062 | 4 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
13. | ALA2349061 | 5 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
14. | ALA2349060 | 6 | INH | 0 | ALA2352358 | Dose-dependent effect | % | Homo sapiens | ||||
15. | ALA2349065 | 1 | IC50 | = | 0.73 | uM | ALA2352358 | 6.14 | nM | Homo sapiens | ||
16. | ALA2349064 | 2 | IC50 | = | 0.71 | uM | ALA2352358 | 6.15 | nM | Homo sapiens | ||
17. | ALA2349063 | 3 | IC50 | = | 0.72 | uM | ALA2352358 | 6.14 | nM | Homo sapiens | ||
18. | ALA2349062 | 4 | IC50 | = | 0.69 | uM | ALA2352358 | 6.16 | nM | Homo sapiens | ||
19. | ALA2349061 | 5 | IC50 | = | 1.1 | uM | ALA2352358 | 5.96 | nM | Homo sapiens | ||
20. | ALA2349060 | 6 | IC50 | = | 2.2 | uM | ALA2352358 | 5.66 | nM | Homo sapiens |