# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | SIAIS178 | 19; SIAIS178 | GI | 0 | ALA4415972 | Active | Homo sapiens | |||||
2. | ALA4439424 | 24 | Activity | 0 | ALA4383466 | Active | Homo sapiens | |||||
3. | ALA4439424 | 24 | Activity | 0 | ALA4383462 | Active | Homo sapiens | |||||
4. | ALA4439424 | 24 | Activity | 0 | ALA4383458 | Active | Homo sapiens | |||||
5. | ALA4519289 | 2 | GI50 | < | 0.001 | uM | ALA4383433 | nM | Homo sapiens | |||
6. | Imatinib (STI571) | 1 | GI50 | = | 0.31 | uM | ALA4383433 | nM | Homo sapiens | |||
7. | ALA4439424 | 24 | GI50 | = | 0.003 | uM | ALA4383433 | nM | Homo sapiens | |||
8. | Axitinib | AG-13736 | GI50 | = | 0.5 | uM | ALA4383433 | nM | Homo sapiens | |||
9. | Dasatinib | 2, BMS-354825 | Activity | 0 | ALA4807714 | Active | Homo sapiens | |||||
10. | Nilotinib (AMN-107) | 38 | IC50 | = | 10 | nM | ALA4316279 | 8.00 | nM | Homo sapiens | ||
11. | ALA4536640 | 69 | IC50 | = | 5 | nM | ALA4316279 | 8.30 | nM | Homo sapiens | ||
12. | ALA4586068 | 62 | IC50 | = | 18 | nM | ALA4316279 | 7.75 | nM | Homo sapiens | ||
13. | ALA4559506 | 48 | IC50 | = | 8 | nM | ALA4316279 | 8.10 | nM | Homo sapiens | ||
14. | ALA4543075 | 44 | IC50 | = | 16 | nM | ALA4316279 | 7.80 | nM | Homo sapiens | ||
15. | ALA4444616 | 42 | IC50 | = | 14 | nM | ALA4316279 | 7.85 | nM | Homo sapiens | ||
16. | Imatinib Mesylate (STI571) | 1, Gleevec | EC50 | = | 0.6 | uM | ALA4155097 | 6.22 | nM | Homo sapiens | ||
17. | ALA4166554 | 5i | EC50 | = | 177.5 | uM | ALA4155097 | nM | Homo sapiens | |||
18. | ALA4163110 | 5e | EC50 | = | 41.7 | uM | ALA4155097 | 4.38 | nM | Homo sapiens | ||
19. | ALA4170635 | 5c | EC50 | = | 57.3 | uM | ALA4155097 | 4.24 | nM | Homo sapiens | ||
20. | ALA4177432 | 1 | EC50 | = | 38.9 | uM | ALA4155097 | 4.41 | nM | Homo sapiens |