# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5267741 | 2 | Activity | 0 | ALA5230031 | Not Active | Homo sapiens | |||||
2. | ALA5286325 | 1 | Activity | 0 | ALA5230031 | Active | Homo sapiens | |||||
3. | ALA2105685 | AMUVATINIB HYDROCHLORIDE | IC50 | = | 27.03 | uM | ALA3992019 | 4.57 | nM | Homo sapiens | ||
4. | ALA2105685 | AMUVATINIB HYDROCHLORIDE | IC50 | = | 66.3 | uM | ALA3992018 | 4.18 | nM | Homo sapiens | ||
5. | ALA2105685 | AMUVATINIB HYDROCHLORIDE | IC50 | = | 7.86 | uM | ALA3992017 | 5.11 | nM | Homo sapiens | ||
6. | BMS-986158 | EZOBRESIB | IC50 | = | 441 | nM | ALA5054352 | 6.36 | nM | Homo sapiens | ||
7. | ALA5268484 | 11; GNE-375 | IC50 | = | 5 | uM | ALA5262606 | 5.30 | nM | Homo sapiens | ||
8. | ALA5268484 | 11; GNE-375 | IC50 | = | 2 | uM | ALA5261773 | 5.70 | nM | Homo sapiens | ||
9. | ALA5270178 | 5 | IC50 | = | 20 | uM | ALA5261773 | 4.70 | nM | Homo sapiens | ||
10. | ALA5282240 | 3 | IC50 | = | 20 | uM | ALA5261773 | 4.70 | nM | Homo sapiens | ||
11. | ALA1641990 | 9 | GI50 | = | 26.303 | uM | ALA1646756 | nM | Homo sapiens | |||
12. | Crizotinib | 14, PF-2341066 | Activity | = | 0.81 | ALA971328 | Homo sapiens | |||||
13. | PD173074 | 12 | Activity | = | 0.85 | ALA971328 | Homo sapiens | |||||
14. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 0.772 | ALA971328 | Homo sapiens | |||||
15. | Imatinib (STI571) | 1 | Activity | = | 0.979 | ALA971328 | Homo sapiens | |||||
16. | Tozasertib | VX-680 | Activity | = | 0.652 | ALA971328 | Homo sapiens | |||||
17. | Neratinib (HKI-272) | 25o (table 3) | Activity | = | 0.879 | ALA971328 | Homo sapiens | |||||
18. | MnTMPyP pentachloride | 5 | Activity | = | 1.007 | ALA971328 | Homo sapiens | |||||
19. | PHA-665752 | PHA-665752 | Activity | = | 0.881 | ALA971328 | Homo sapiens | |||||
20. | Sunitinib | 12b | Activity | = | 1.01 | ALA971328 | Homo sapiens |