1. | ALA2072537 | A | Stability in human plasma assessed as compound remaining at 1 hr | Homo sapiens | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | cell-free format | Scientific Literature |
2. | ALA2072538 | A | Protein binding in mouse | Mus musculus | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | organism-based format | Scientific Literature |
3. | ALA2072539 | A | Protein binding in rat | Rattus norvegicus | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | organism-based format | Scientific Literature |
4. | ALA2072540 | A | Protein binding in human | Homo sapiens | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | organism-based format | Scientific Literature |
5. | ALA2072541 | P | Solubility of the compound at pH 1-9 | | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | small-molecule physicochemical format | Scientific Literature |
6. | ALA2072542 | A | Metabolic stability in rat liver microsomes assessed as compound remaining at 1 hr | Rattus norvegicus | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | microsome format | Scientific Literature |
7. | ALA2072543 | A | Metabolic stability in mouse liver microsomes assessed as compound remaining at 1 hr | Mus musculus | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | microsome format | Scientific Literature |
8. | ALA2072544 | A | Metabolic stability in dog liver microsomes assessed as compound remaining at 1 hr | Canis lupus familiaris | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | microsome format | Scientific Literature |
9. | ALA2072545 | A | Metabolic stability in human liver microsomes assessed as compound remaining at 1 hr | Homo sapiens | 1 | 22850208 10.1016/j.bmcl.2012.07.019 | microsome format | Scientific Literature |
10. | ALA2072546 | B | Displacement of [3H](+)-pentazocine from sigma1 receptor in guinea pig brain homogenate | Cavia porcellus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
11. | ALA2072547 | B | Displacement of [3H]DTG from sigma2 receptor in rat liver homogenate in presence of (+)-pentazocine | Rattus norvegicus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
12. | ALA2072548 | B | Selectivity ratio of Ki for rat sigma2 receptor to Ki for guinea pig sigma1 receptor | | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | assay format | Scientific Literature |
13. | ALA2072549 | B | Binding affinity to sigma1 receptor in guinea pig brain homogenate | Cavia porcellus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
14. | ALA2072550 | B | Binding affinity to sigma2 receptor in guinea pig brain homogenate | Cavia porcellus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
15. | ALA2072551 | B | Binding affinity to sigma1 receptor | Homo sapiens | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | single protein format | Scientific Literature |
16. | ALA2072552 | B | Binding affinity to sigma2 receptor | Homo sapiens | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | assay format | Scientific Literature |
17. | ALA2072553 | B | Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenate after 120 mins | Rattus norvegicus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
18. | ALA2072554 | B | Displacement of [3H]DTG from sigma2 receptor in rat brain homogenate in presence of (+)-pentazocine after 120 mins | Rattus norvegicus | 1 | 22850210 10.1016/j.bmcl.2012.07.026 | tissue-based format | Scientific Literature |
19. | ALA2072555 | F | Insecticidal activity against 5th instar nymph of Dysdercus koenigii assessed as mortality per nymph | Dysdercus koenigii | 1 | 22850211 10.1016/j.bmcl.2012.07.017 | assay format | Scientific Literature |
20. | ALA2072556 | F | Insecticidal activity against 5th instar nymph of Dysdercus koenigii assessed as smaller body size at 20 and 50 ug/nymph | Dysdercus koenigii | 1 | 22850211 10.1016/j.bmcl.2012.07.017 | assay format | Scientific Literature |