| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1794424 | F | PUBCHEM_BIOASSAY: qHTS Assay for Inhibitors of Mammalian Selenoprotein Thioredoxin Reductase 1 (TrxR1): qHTS. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID488771] | 30,565 | assay format | PubChem BioAssays | |||
| 2. | ALA1117927 | B | Inhibition of ROCK2 | 30 | single protein format | Scientific Literature | |||
| 3. | ALA1117929 | B | Inhibition of ROCK1 | 8 | single protein format | Scientific Literature | |||
| 4. | ALA1117930 | B | Inhibition of Prkce | 8 | single protein format | Scientific Literature | |||
| 5. | ALA1117931 | B | Inhibition of DMPK | 8 | single protein format | Scientific Literature | |||
| 6. | ALA1117932 | B | Inhibition of CDc42 | 8 | single protein format | Scientific Literature | |||
| 7. | ALA1117933 | B | Inhibition of Prkcl2 | 8 | single protein format | Scientific Literature | |||
| 8. | ALA1118080 | A | Metabolic stability in rat liver microsomes | Rattus norvegicus | 4 | microsome format | Scientific Literature | ||
| 9. | ALA1118081 | A | Metabolic stability in human liver microsomes | Homo sapiens | 4 | microsome format | Scientific Literature | ||
| 10. | ALA1118082 | P | Solubility at pH 7.4 | 4 | small-molecule physicochemical format | Scientific Literature | |||
| 11. | ALA1118083 | A | Clearance in rat at 1 mg/kg, iv and 10 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 12. | ALA1118084 | A | Half life in rat at 1 mg/kg, iv and 10 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 13. | ALA1118085 | A | AUC in rat at 1 mg/kg, iv and 10 mg/kg, po | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 14. | ALA1118086 | A | Oral bioavailability in rat at 10 mg/kg | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 15. | ALA1118087 | A | Inhibition of CYP1A2 | 4 | single protein format | Scientific Literature | |||
| 16. | ALA1118088 | A | Inhibition of CYP2D6 | 2 | single protein format | Scientific Literature | |||
| 17. | ALA1118089 | A | Inhibition of CYP3A4 | 2 | single protein format | Scientific Literature | |||
| 18. | ALA1118090 | B | Inhibition of human ERG | 4 | single protein format | Scientific Literature | |||
| 19. | ALA1118091 | F | Cytotoxicity against human HeLa cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 20. | ALA1118093 | F | Vasodilatory activity in Sprague-Dawley rat assessed as inhibition of aortic ring contraction | Rattus norvegicus | 4 | organism-based format | Scientific Literature |
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