#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA1648234	Binding	Displacement of [125I]glucagon from human GCGR expressed in CHO cells	Homo sapiens	41	ALA1641377	cell-based format	Scientific Literature
2.	ALA1648235	Functional	Antagonist activity at human GCGR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation	Homo sapiens	41	ALA1641377	cell-based format	Scientific Literature
3.	ALA1648236	Functional	Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation	Homo sapiens	19	ALA1641377	cell-based format	Scientific Literature
4.	ALA1648240	Functional	Antidiabetic activity in transgenic mouse expressing human GCGR assessed as inhibition of glucagon-induced blood glucose excursion at 30 mg/kg, po administered 3 hrs before glucagon challenge measured after 48 mins	Mus musculus	1	ALA1641377	organism-based format	Scientific Literature
5.	ALA1648241	Functional	Antidiabetic activity in transgenic mouse expressing human GCGR assessed as inhibition of glucagon-induced blood glucose excursion at 30 mg/kg, po administered 60 mins before glucagon challenge measured after 48 mins	Mus musculus	4	ALA1641377	organism-based format	Scientific Literature
6.	ALA1648242	Functional	Antidiabetic activity in transgenic mouse expressing human GCGR assessed as inhibition of glucagon-induced blood glucose excursion at 10 mg/kg, po administered 60 mins before glucagon challenge measured after 48 mins	Mus musculus	5	ALA1641377	organism-based format	Scientific Literature
7.	ALA1648243	ADME	Drug level in blood of transgenic mouse expressing human GCGR at 10 mg/kg, po after 45 mins	Mus musculus	1	ALA1641377	organism-based format	Scientific Literature
8.	ALA1648244	ADME	Drug level in blood of transgenic mouse expressing human GCGR at 10 mg/kg, po after 120 mins	Mus musculus	1	ALA1641377	organism-based format	Scientific Literature
9.	ALA1648245	ADME	Drug level in blood of transgenic mouse expressing human GCGR at 30 mg/kg, po after 45 mins	Mus musculus	1	ALA1641377	organism-based format	Scientific Literature
10.	ALA1648246	ADME	Drug level in blood of transgenic mouse expressing human GCGR at 30 mg/kg, po after 120 mins	Mus musculus	1	ALA1641377	organism-based format	Scientific Literature
11.	ALA1648248	Functional	Antagonist activity at human GLP1R expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation	Homo sapiens	1	ALA1641377	cell-based format	Scientific Literature
12.	ALA1648771	Functional	Antagonist activity at human PACAPR1 expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation	Homo sapiens	1	ALA1641377	cell-based format	Scientific Literature
13.	ALA1648772	Binding	Inhibition of human ERG	Homo sapiens	1	ALA1641377	single protein format	Scientific Literature
14.	ALA1648773	Binding	Binding affinity to human sodium channel up to 10 uM	Homo sapiens	1	ALA1641377	assay format	Scientific Literature
15.	ALA1648774	Binding	Binding affinity to DLZ-sensitive rabbit calcium channel up to 10 uM	Oryctolagus cuniculus	1	ALA1641377	assay format	Scientific Literature
16.	ALA1648775	Toxicity	Cardiotoxicity in dog assessed as effect on cardiovascular parameters at 1 to 10 mg/kg, iv after 30 mins	Canis lupus familiaris	1	ALA1641377	organism-based format	Scientific Literature
17.	ALA1648776	ADME	Plasma concentration in dog at 1 to 10 mg/kg, iv after 30 mins	Canis lupus familiaris	1	ALA1641377	organism-based format	Scientific Literature
18.	ALA1648777	ADME	Inhibition of CYP2D6		1	ALA1641377	single protein format	Scientific Literature
19.	ALA1648778	ADME	Inhibition of CYP3A4		1	ALA1641377	single protein format	Scientific Literature
20.	ALA1648779	ADME	Inhibition of CYP2C8		1	ALA1641377	single protein format	Scientific Literature