| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1679250 | B | Displacement of [3H]-ZM241385 from human adenosine A2A receptor expressed in high five cells after 30 mins by scintillation counting | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 2. | ALA1679251 | B | Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells after 30 mins by scintillation counting | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 3. | ALA1679257 | A | Inhibition of recombinant CYP1A2 after 28 mins | 8 | single protein format | Scientific Literature | |||
| 4. | ALA1679258 | A | Inhibition of recombinant CYP2C9 after 45 mins | 7 | single protein format | Scientific Literature | |||
| 5. | ALA1679259 | A | Inhibition of recombinant CYP2C19 after 45 mins | 8 | single protein format | Scientific Literature | |||
| 6. | ALA1679408 | A | Inhibition of recombinant CYP2D6 after 45 mins | 8 | single protein format | Scientific Literature | |||
| 7. | ALA1679409 | A | Inhibition of recombinant CYP3A4 after 30 mins | 7 | single protein format | Scientific Literature | |||
| 8. | ALA1679414 | B | Selectivity ratio of Ki for human adenosine A1 receptor to Ki for human adenosine A2A receptor | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 9. | ALA1679415 | F | Antagonist activity at human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA1679416 | B | Displacement of [3H]-MRS1754 from human recombinant adenosine A2B receptor expressed in HEK293 cells after 60 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA1679417 | B | Displacement of [3H]-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO-K1 cells after 60 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA1679418 | B | Displacement of [3H]-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO-K1 cells at 10 uM after 60 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA1679419 | B | Selectivity ratio of Ki for human adenosine A2B receptor to Ki for human adenosine A2A receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA1679420 | B | Selectivity ratio of Ki for human adenosine A3 receptor to Ki for human adenosine A2A receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA1679421 | A | Intrinsic clearance in rat hepatocytes at 0.2 uM after 60 mins | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA1679422 | A | Intrinsic clearance in dog hepatocytes at 0.2 uM after 60 mins | Canis lupus familiaris | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA1679423 | A | Intrinsic clearance in human hepatocytes at 0.2 uM after 60 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA1679424 | A | Apparent permeability from apical to basolateral side in human Caco2 cells at 1 uM after 21 to 28 days | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA1679425 | A | Apparent permeability from basolateral to apical side in human Caco2 cells at 1 uM after 21 to 28 days | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA1679426 | A | Protein binding in rat serum at 1 uM after 60 mins by LC/MS-MS | Rattus norvegicus | 1 | cell-free format | Scientific Literature |
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