# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1680281 | Binding | Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin (6-14) from human BRS-3 | Homo sapiens | 6 | ALA1671827 | single protein format | Scientific Literature | |
2. | ALA1680282 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
3. | ALA1680283 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay relative to dY peptide | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
4. | ALA1680284 | ADME | Half life in rat liver microsomes | Rattus norvegicus | 8 | ALA1671827 | microsome format | Scientific Literature | |
5. | ALA1680287 | Binding | Activation of human PXR | Homo sapiens | 2 | ALA1671827 | single protein format | Scientific Literature | |
6. | ALA1680289 | Binding | Binding affinity to human ERG | Homo sapiens | 3 | ALA1671827 | single protein format | Scientific Literature | |
7. | ALA1680290 | ADME | Plasma clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 6 | ALA1671827 | organism-based format | Scientific Literature | |
8. | ALA1680291 | ADME | Faction unbound in human plasma at 1 uM | Homo sapiens | 6 | ALA1671827 | cell-free format | Scientific Literature | |
9. | ALA1680292 | ADME | Fraction unbound in rat plasma at 1 uM | Rattus norvegicus | 6 | ALA1671827 | cell-free format | Scientific Literature | |
10. | ALA1681379 | Binding | Inhibition of human NMBR | Homo sapiens | 1 | ALA1671827 | single protein format | Scientific Literature | |
11. | ALA1681380 | Binding | Inhibition of human GRPR | Homo sapiens | 1 | ALA1671827 | single protein format | Scientific Literature | |
12. | ALA1681381 | Binding | Inhibition of human calcium channel diltiazem binding site | Homo sapiens | 2 | ALA1671827 | assay format | Scientific Literature |