| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1686104 | B | Inhibition of human CCR2 by human whole blood assay | Homo sapiens | 1 | ALA1681706 | tissue-based format | Scientific Literature | |
| 2. | ALA1686105 | B | Displacement of [125I]MCP1 from human CCR2 by human whole cell binding assay | Homo sapiens | 1 | ALA1681706 | single protein format | Scientific Literature | |
| 3. | ALA1686106 | A | Half life in human liver microsomes at 1 uM | Homo sapiens | 33 | ALA1681706 | microsome format | Scientific Literature | |
| 4. | ALA1686112 | B | Displacement of dofetilide from human ERG | Homo sapiens | 1 | ALA1681706 | single protein format | Scientific Literature | |
| 5. | ALA1685777 | B | Displacement of [125I]MCP1 from human CCR2 after 30 mins by gamma counting | Homo sapiens | 35 | ALA1681668 | single protein format | Scientific Literature | |
| 6. | ALA1685778 | F | Antagonist activity at human CCR2 in human PBMC assessed as inhibition of MCP1-induced chemotaxis after 30 mins | Homo sapiens | 8 | ALA1681668 | assay format | Scientific Literature | |
| 7. | ALA1685779 | B | Displacement of labeled MIP-1beta from human CCR5 receptor | Homo sapiens | 19 | ALA1681668 | single protein format | Scientific Literature | |
| 8. | ALA1685780 | B | Displacement of MCP-Alexa 488 from CCR2 in human whole blood after 5 mins by flow cytometry | Homo sapiens | 11 | ALA1681668 | single protein format | Scientific Literature | |
| 9. | ALA1685781 | F | Antagonist activity at human CCR5 receptor by chemotaxis assay | Homo sapiens | 2 | ALA1681668 | assay format | Scientific Literature | |
| 10. | ALA1685782 | B | Binding affinity to mouse CCR2 | Mus musculus | 1 | ALA1681668 | single protein format | Scientific Literature | |
| 11. | ALA1685783 | B | Binding affinity to rat CCR2 | Rattus norvegicus | 1 | ALA1681668 | single protein format | Scientific Literature | |
| 12. | ALA1685784 | B | Binding affinity to cynomolgus monkey CCR2 | Macaca fascicularis | 1 | ALA1681668 | assay format | Scientific Literature | |
| 13. | ALA1685785 | B | Binding affinity to dog CCR2 | Canis lupus familiaris | 1 | ALA1681668 | assay format | Scientific Literature | |
| 14. | ALA1685786 | B | Binding affinity to mouse CCR5 | Mus musculus | 1 | ALA1681668 | single protein format | Scientific Literature | |
| 15. | ALA1685787 | B | Binding affinity to cynomolgus monkey CCR5 | Macaca fascicularis | 1 | ALA1681668 | assay format | Scientific Literature | |
| 16. | ALA1685788 | A | Inhibition of human CYP3A4 | Homo sapiens | 1 | ALA1681668 | single protein format | Scientific Literature | |
| 17. | ALA1685789 | A | Inhibition of human CYP2D6 | Homo sapiens | 1 | ALA1681668 | single protein format | Scientific Literature | |
| 18. | ALA1685790 | B | Inhibition of human ERG by patch clamp assay | Homo sapiens | 1 | ALA1681668 | assay format | Scientific Literature | |
| 19. | ALA1686155 | A | Permeability of the compound across human Caco2 cells | Homo sapiens | 1 | ALA1681668 | cell-based format | Scientific Literature | |
| 20. | ALA1686156 | A | Fraction unbound in human plasma | Homo sapiens | 1 | ALA1681668 | cell-free format | Scientific Literature |
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