| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1686343 | Binding | Inhibition of human PKD1 by TR-FRET assay | Homo sapiens | 27 | ALA1681675 | single protein format | Scientific Literature | |
| 2. | ALA1686344 | ADME | Half life in rat liver microsomes | Rattus norvegicus | 26 | ALA1681675 | microsome format | Scientific Literature | |
| 3. | ALA1686345 | Physicochemical | Solubility of the compound | 26 | ALA1681675 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA1686346 | Binding | Inhibition of human PKD2 | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 5. | ALA1686347 | Binding | Inhibition of human PKD3 | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 6. | ALA1686348 | Binding | Inhibition of human PKD2 at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 7. | ALA1686349 | Binding | Inhibition of human CaMK1delta at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 8. | ALA1686350 | Binding | Inhibition of rat CaMK2alpha at 1 uM | Rattus norvegicus | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 9. | ALA1686351 | Binding | Inhibition of human CaMK2beta at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 10. | ALA1686352 | Binding | Inhibition of human CaMK2delta at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 11. | ALA1686353 | Binding | Inhibition of human CaMK4 at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 12. | ALA1686354 | Binding | Inhibition of human MARK1 at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 13. | ALA1686355 | Binding | Inhibition of human SIK at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 14. | ALA1686356 | Binding | Inhibition of human GRK5 at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 15. | ALA1686357 | Binding | Inhibition of human PKCdelta at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 16. | ALA1686358 | Binding | Inhibition of human PKCepsilon at 1 uM | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 17. | ALA1686359 | Binding | Inhibition of human CaMK2delta | Homo sapiens | 1 | ALA1681675 | single protein format | Scientific Literature | |
| 18. | ALA1686360 | Binding | Selectivity ratio, ratio of IC50 for human PKD1 to IC50 for human PKD2 | Homo sapiens | 1 | ALA1681675 | assay format | Scientific Literature | |
| 19. | ALA1686361 | Binding | Selectivity ratio, ratio of IC50 for human PKD1 to IC50 for human PKD3 | Homo sapiens | 1 | ALA1681675 | assay format | Scientific Literature | |
| 20. | ALA1686362 | Binding | Inhibition of PKD1 in rat neonatal ventricular myocytes expressing GFP-HDAC5 assessed as inhibition of phosphorylation-dependent HDAC5 nuclear export | Rattus norvegicus | 5 | ALA1681675 | cell-based format | Scientific Literature |
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