| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1810552 | B | Displacement of [3H]AVP from human V1A receptor expressed in CHO cells | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 2. | ALA1810823 | B | Displacement of [3H]AVP from rat V1A receptor expressed in CHO cells | Rattus norvegicus | 21 | cell-based format | Scientific Literature | ||
| 3. | ALA1810825 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 27 | microsome format | Scientific Literature | ||
| 4. | ALA1810826 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 27 | microsome format | Scientific Literature | ||
| 5. | ALA1810827 | A | Apparent permeability of the compound from apical to basolateral side of human Caco2 cells | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
| 6. | ALA1810828 | A | Efflux ratio of permeability from apical to basolateral over basolateral to apical side in human Caco2 cells | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
| 7. | ALA1776763 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 11 | microsome format | Scientific Literature | ||
| 8. | ALA1776930 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 10 | microsome format | Scientific Literature | ||
| 9. | ALA1776931 | B | Displacement of [3H]AVP from human V1A receptor expressed in CHO cells | Homo sapiens | 41 | cell-based format | Scientific Literature | ||
| 10. | ALA1776932 | B | Displacement of [3H]AVP from rat V1A receptor expressed in CHO cells | Rattus norvegicus | 9 | cell-based format | Scientific Literature | ||
| 11. | ALA1776935 | A | Oral bioavailability in po dosed Wistar rat at 10 mg/kg | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 12. | ALA1776936 | A | Half life in Wistar rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 13. | ALA1776937 | A | Cmax in Wistar rat at 10 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 14. | ALA1776938 | A | Tmax in Wistar rat at 10 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 15. | ALA1776939 | A | Volume of distribution at steady state in Wistar rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 16. | ALA1776940 | A | Plasma clearance in Wistar rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 17. | ALA1776941 | F | Antagonist activity at human V1A receptor expressed in CHO cells assessed as inhibition of AVP-induced intracellular calcium release | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA1776942 | B | Displacement of [3H]dofetilide from human ERG expressed in HEK293 cells | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 19. | ALA1776943 | B | Displacement of [3H]AVP from human V1B receptor expressed in CHO cells | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 20. | ALA1776944 | B | Displacement of [3H]AVP from human V2 receptor expressed in CHO cells | Homo sapiens | 2 | cell-based format | Scientific Literature |
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