| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1781790 | B | Inhibition of human SGLT2 expressed in CHO cells assessed as inhibition of [14C]-Glucose uptake using [14C]-methyl glucopyranoside after 60 mins by microbeta plate counting | Homo sapiens | 33 | ALA1777714 | cell-based format | Scientific Literature | |
| 2. | ALA1781791 | A | Metabolic stability in rat liver microsomes assessed as compound remaining at 1 uM after 30 mins by liquid chromatography/mass spectrometry analysis | Rattus norvegicus | 26 | ALA1777714 | microsome format | Scientific Literature | |
| 3. | ALA1781792 | A | Metabolic stability in human liver microsomes assessed as compound remaining at 1 uM after 30 mins by liquid chromatography/mass spectrometry analysis | Homo sapiens | 26 | ALA1777714 | microsome format | Scientific Literature | |
| 4. | ALA1781793 | P | Solubility of the compound in phosphate buffered saline | 10 | ALA1777714 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA1781796 | B | Inhibition of human SGLT1 | Homo sapiens | 3 | ALA1777714 | single protein format | Scientific Literature | |
| 6. | ALA1781797 | B | Inhibition of rat SGLT2 | Rattus norvegicus | 2 | ALA1777714 | single protein format | Scientific Literature | |
| 7. | ALA1781798 | A | Cmax in rat at 100 mg/kg, sc | Rattus norvegicus | 1 | ALA1777714 | organism-based format | Scientific Literature | |
| 8. | ALA1781800 | A | AUC (0 to 24 hrs) in rat at 100 mg/kg, sc | Rattus norvegicus | 1 | ALA1777714 | organism-based format | Scientific Literature | |
| 9. | ALA1780641 | A | Tmax in rat at 100 mg/kg, sc | Rattus norvegicus | 1 | ALA1777714 | organism-based format | Scientific Literature | |
| 10. | ALA1780643 | A | Fraction unbound in rat plasma at 100 mg/kg, sc | Rattus norvegicus | 1 | ALA1777714 | organism-based format | Scientific Literature |
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