| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1787313 | B | Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as reduction in [14C]-alpha-methylglucopyranoside uptake after 2 hrs by liquid scintillation counting | Homo sapiens | 21 | ALA1781960 | cell-based format | Scientific Literature | |
| 2. | ALA3110555 | B | Selectivity ratio of IC50 for human SGLT1 to IC50 for human SGLT2 | Homo sapiens | 3 | ALA3108724 | assay format | Scientific Literature | |
| 3. | ALA3110556 | T | Toxicity in high-fat diet-fed KK/Ta Jcl mouse assessed as effect on food intake at 3 mg/kg, po | Mus musculus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 4. | ALA3110557 | F | Antihyperglycemic activity in high-fat diet-fed KK/Ta Jcl mouse assessed as reduction in blood glucose level at 3 mg/kg, po measured at 24 hrs | Mus musculus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 5. | ALA3110558 | A | Metabolic stability in monkey intestinal microsomes assessed as compound hydrolysis by HPLC analysis | Macaca mulatta | 1 | ALA3108724 | assay format | Scientific Literature | |
| 6. | ALA3110559 | A | Metabolic stability in dog intestinal microsomes assessed as compound hydrolysis by HPLC analysis | Canis lupus familiaris | 1 | ALA3108724 | assay format | Scientific Literature | |
| 7. | ALA3110560 | A | Metabolic stability in rat intestinal microsomes assessed as compound hydrolysis by HPLC analysis | Rattus norvegicus | 1 | ALA3108724 | assay format | Scientific Literature | |
| 8. | ALA3110561 | A | Metabolic stability in human intestinal microsomes assessed as compound hydrolysis by HPLC analysis | Homo sapiens | 1 | ALA3108724 | assay format | Scientific Literature | |
| 9. | ALA3110562 | A | Intrinsic clearance in monkey intestinal microsomes after 30 mins | Macaca mulatta | 1 | ALA3108724 | assay format | Scientific Literature | |
| 10. | ALA3110563 | A | Intrinsic clearance in rat intestinal microsomes after 30 mins | Rattus norvegicus | 1 | ALA3108724 | assay format | Scientific Literature | |
| 11. | ALA3110564 | A | Intrinsic clearance in dog intestinal microsomes after 30 mins | Canis lupus familiaris | 1 | ALA3108724 | assay format | Scientific Literature | |
| 12. | ALA3110565 | A | Intrinsic clearance in human intestinal microsomes after 30 mins | Homo sapiens | 1 | ALA3108724 | assay format | Scientific Literature | |
| 13. | ALA3110566 | A | Oral bioavailability in Sprague-Dawley rat at 10 mg/kg | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 14. | ALA3110567 | A | Volume of distribution at steady state in Sprague-Dawley rat at 3 mg/kg, iv | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 15. | ALA3110568 | A | Total clearance in Sprague-Dawley rat at 3 mg/kg, iv | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 16. | ALA3110569 | A | Half life in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 17. | ALA3110570 | A | Half life in Sprague-Dawley rat at 3 mg/kg, iv | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 18. | ALA3110571 | A | AUC (0 to infinity) in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 19. | ALA3110572 | A | AUC (0 to infinity) in Sprague-Dawley rat at 3 mg/kg, iv | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature | |
| 20. | ALA3110573 | A | Tmax in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA3108724 | organism-based format | Scientific Literature |
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