# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA960986 | B | Inhibition of human PLK1 kinase domain expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay | Homo sapiens | 16 | ALA1153318 | cell-based format | Scientific Literature | |
2. | ALA960987 | B | Inhibition of full length human PLK3 expressed in baculovirus-infected Trichoplusia ni cells by scintillation proximity assay | Homo sapiens | 16 | ALA1153318 | cell-based format | Scientific Literature | |
3. | ALA960988 | F | Antiproliferative activity against human HCT116 cells after 72 hrs by luminescence-based cell viability assay | Homo sapiens | 15 | ALA1153318 | cell-based format | Scientific Literature | |
4. | ALA960989 | P | Solubility in 0.05 M phosphate buffer at 200 uM at pH 7.4 after 15 mins by HPLC | 13 | ALA1153318 | small-molecule physicochemical format | Scientific Literature | ||
5. | ALA960990 | A | Protein binding in human plasma at 2000 ng/mL after 6 hrs by equilibrium dialysis method | Homo sapiens | 11 | ALA1153318 | cell-free format | Scientific Literature | |
6. | ALA1961874 | B | GSK_PKIS: AKT1 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
7. | ALA1961875 | B | GSK_PKIS: AKT1 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
8. | ALA1961876 | B | GSK_PKIS: AKT2 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
9. | ALA1961877 | B | GSK_PKIS: AKT2 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
10. | ALA1961878 | B | GSK_PKIS: AKT3 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
11. | ALA1961879 | B | GSK_PKIS: AKT3 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
12. | ALA1961880 | B | GSK_PKIS: GRK6 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
13. | ALA1961881 | B | GSK_PKIS: GRK6 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
14. | ALA1961882 | B | GSK_PKIS: GRK7 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
15. | ALA1961883 | B | GSK_PKIS: GRK7 mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
16. | ALA1961884 | B | GSK_PKIS: MRCKA mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
17. | ALA1961885 | B | GSK_PKIS: MRCKA mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
18. | ALA1961886 | B | GSK_PKIS: MRCKB mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
19. | ALA1961887 | B | GSK_PKIS: MRCKB mean inhibition at 1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set | ||
20. | ALA1961888 | B | GSK_PKIS: MSK1 mean inhibition at 0.1 uM [Nanosyn] | 366 | ALA1961873 | single protein format | GSK Published Kinase Inhibitor Set |