| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1798505 | B | Competitive inhibition of p300 HAT | 1 | single protein format | Scientific Literature | |||
| 2. | ALA3391521 | B | Competitive inhibition of p300 (unknown origin) using acetyl CoA as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3778079 | B | Inhibition of FLAG-tagged p300 (1195 to 1673 residues) (unknown origin) expressed in competent Escherichia coli BL21-CodonPlus(DE3)-RIL cells using histone H4 substrate incubated for 10 mins by scintillation counting method in presence of [14C]acetyl-CoA | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA3779177 | B | Inhibition of PCAF (unknown origin) using H4-15 peptide substrate at 10 uM incubated for 10 mins by radiometric filter binding assay in presence of [14C]acetyl-CoA relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA3779180 | B | Inhibition of yeast GCN5 using histone H3 substrate at 10 uM incubated for 2 to 4 mins by SDS-PAGE based autoradiography in presence of [14C]acetyl-CoA relative to control | Saccharomyces cerevisiae | 1 | assay format | Scientific Literature | ||
| 6. | ALA3779392 | B | Inhibition of synthetic VMA-tagged p300 (1287 to 1652 residues) (unknown origin) expressed in Escherichia coli BL21(RIL)-DE3 cells using H4-15 peptide substrate incubated for 10 mins by radiometric filter binding assay in presence of [14C]acetyl-CoA | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA3779393 | B | Inhibition of synthetic VMA-tagged p300 (1287 to 1652 residues) (unknown origin) expressed in Escherichia coli BL21(RIL)-DE3 cells using H4-15 peptide substrate at 10 uM incubated for 10 mins by radiometric filter binding assay in presence of [14C]acetyl-CoA relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA3779394 | B | Inhibition of yeast RTT109 using histone H3 substrate at 10 uM incubated for 2 to 4 mins by SDS-PAGE based autoradiography in presence of [14C]acetyl-CoA relative to control | Saccharomyces cerevisiae | 1 | assay format | Scientific Literature | ||
| 9. | ALA3779395 | B | Inhibition of yeast YJW458 TAP-tagged SAS2 expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL cells using histone H3 as substrate at 10 uM incubated for 2 to 4 mins by SDS-PAGE based autoradiography in presence of [14C]acetyl-CoA relative to control | Saccharomyces cerevisiae | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA3779396 | B | Inhibition of human MOZ using histone H3 substrate at 10 uM incubated for 2 to 4 mins by SDS-PAGE based autoradiography in presence of [14C]acetyl-CoA relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA3803991 | B | Inhibition of porcine brain tubulin polymerization assessed as decrease in rate of microtubule formation incubated up to 1 hr by fluorescence analysis | Sus scrofa | 1 | assay format | Scientific Literature | ||
| 12. | ALA3803992 | B | Inhibition of recombinant P300 (1195 to 1662 residues) (unknown origin) using FITC-histone H4 as substrate incubated for 10 mins by microfluidic electrophoresis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA3803993 | B | Inhibition of recombinant P300 (1195 to 1662 residues) (unknown origin) using FITC-histone H4 as substrate incubated for 10 mins by microfluidic electrophoresis in presence of BSA | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3803994 | B | Inhibition of recombinant P300 (1195 to 1662 residues) (unknown origin) using FITC-histone H4 as substrate incubated for 10 mins by microfluidic electrophoresis in presence of DTT | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3803995 | B | Inhibition of recombinant P300 (1195 to 1662 residues) (unknown origin) using FITC-histone H4 as substrate incubated for 10 mins by microfluidic electrophoresis in presence of DTT and BSA | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA3803996 | B | Inhibition of P300 in human HepG2 cells using H3K27 as substrate at 20 to 40 uM incubated for 24 hrs by Western blot analysis in presence of BSA | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA3803997 | B | Inhibition of recombinant P300 catalytic domain (1284 to 1673 residues) (unknown origin) using FITC- histone H4 peptide (1 to 19 residues) as substrate by electrophoretic mobility shift assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 18. | ALA4325422 | B | Inhibition of VMA intein chitin binding domain-fused P300 (unknown origin) (1287 to 1652 residues) expressed in Escherichia coli BL21(RIL)-DE3 cells using [12C]-acetyl-CoA/[14C]-acetyl-CoA as substrate preincubated for 10 mins followed by substrate addition and measured after 10 mins by phosphor imaging analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4327287 | F | Antiplasmodial activity against asynchronous form of Plasmodium falciparum 3D7 infected in human erythrocytes assessed as parasite growth inhibition at 10 uM after 48 hrs by SYBR green1 staining based flow cytometry relative to control | Plasmodium falciparum | 51 | organism-based format | Scientific Literature | ||
| 20. | ALA4327288 | F | Antiplasmodial activity against asynchronous form of Plasmodium falciparum 3D7 infected in human erythrocytes assessed as parasite growth inhibition after 48 hrs by SYBR green1 staining based flow cytometry | Plasmodium falciparum | 52 | organism-based format | Scientific Literature |
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