# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1805099 | B | Inhibition of rat recombinant GST-tagged DYRK1A using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation counting | Rattus norvegicus | 39 | ALA1800025 | single protein format | Scientific Literature | |
2. | ALA1805100 | B | Inhibition of human recombinant GST-tagged DYRK2 using KKISGRLSPIMTEQ as substrate and [gamma32]-ATP after 30 mins by scintillation counting | Homo sapiens | 39 | ALA1800025 | single protein format | Scientific Literature | |
3. | ALA1805101 | B | Inhibition of mouse recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrate | Mus musculus | 38 | ALA1800025 | single protein format | Scientific Literature | |
4. | ALA1805102 | B | Inhibition of mouse recombinant GST-tagged CLK3 using GRSRSRSRSRSR as substrate | Mus musculus | 38 | ALA1800025 | single protein format | Scientific Literature | |
5. | ALA1805103 | B | Inhibition of human recombinant CDK5/p25 | Homo sapiens | 35 | ALA1800025 | protein complex format | Scientific Literature | |
6. | ALA1805106 | B | Inhibition of human recombinant Pim1 | Homo sapiens | 41 | ALA1800025 | single protein format | Scientific Literature | |
7. | ALA1805112 | B | Inhibition of pig brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrate at 10 uM | Sus scrofa | 40 | ALA1800025 | assay format | Scientific Literature | |
8. | ALA1805113 | B | Inhibition of pig brain CK1 delta/epsilon using RRKHAAIGpSAYSITA as substrate at 10 uM | Sus scrofa | 39 | ALA1800025 | assay format | Scientific Literature | |
9. | ALA5127367 | B | Inhibition of porcine brain GSK-3alpha/beta using YRRAAVPPSPSLSRHSSPHQpSEDEEE as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Sus scrofa | 49 | ALA5126517 | tissue-based format | Scientific Literature | |
10. | ALA5127369 | B | Inhibition of GST-fused mouse recombinant CLK4 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Mus musculus | 60 | ALA5126517 | assay format | Scientific Literature | |
11. | ALA5127372 | B | Inhibition of GST-fused mouse recombinant CLK3 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Mus musculus | 50 | ALA5126517 | assay format | Scientific Literature | |
12. | ALA5127373 | B | Inhibition of GST-fused mouse recombinant CLK1 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Mus musculus | 60 | ALA5126517 | assay format | Scientific Literature | |
13. | ALA5127375 | B | Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Mus musculus | 57 | ALA5126517 | assay format | Scientific Literature | |
14. | ALA5127377 | B | Inhibition of GST-fused human recombinant DYRK1A expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 61 | ALA5126517 | assay format | Scientific Literature | |
15. | ALA5127379 | B | Inhibition of GST-fused human recombinant DYRK1B expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 58 | ALA5126517 | assay format | Scientific Literature | |
16. | ALA5127381 | B | Inhibition of GST-fused human recombinant DYRK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 59 | ALA5126517 | assay format | Scientific Literature | |
17. | ALA5127383 | B | Inhibition of GST-fused human recombinant DYRK3 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 53 | ALA5126517 | assay format | Scientific Literature | |
18. | ALA5127386 | B | Inhibition of human recombinant Pim1 expressed in Escherichia coli using histone H1 as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 52 | ALA5126517 | assay format | Scientific Literature | |
19. | ALA5127388 | B | Inhibition of human recombinant CK2 using RRRDDDSDDD peptide as substrate incubated for 30 mins in presence of ATP by scintillation counting method | Homo sapiens | 43 | ALA5126517 | protein format | Scientific Literature | |
20. | ALA5127391 | F | Neuroprotective activity against glutamate-induced cell death in mouse HT-22 cells treated for 24 hrs by MTS assay | Mus musculus | 41 | ALA5126517 | cell-based format | Scientific Literature |