| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1832655 | B | Inhibition of STAT3 in mouse NIH3T3/vSrc nuclear extract assessed as disruption of the Stat3-DNA complex pre-incubated for 30 mins by EMSA analysis | Mus musculus | 16 | ALA1828629 | single protein format | Scientific Literature | |
| 2. | ALA1832656 | B | Inhibition of STAT3 using fluorescent probe 5-carboxyfluorescein-GpYLPQTV-NH2 after 15 mins by fluorescence polarisation assay | 10 | ALA1828629 | single protein format | Scientific Literature | ||
| 3. | ALA3227583 | B | Mixed inhibition of human GST-tagged PTP1B catalytic domain assessed as rate of DiFMUP hydrolysis by lineweaver-burk plot analysis | Homo sapiens | 1 | ALA3217656 | single protein format | Scientific Literature | |
| 4. | ALA3226166 | A | Cytotoxicity against Chinese hamster CHO cells overexpressing IR assessed as slight reduction in cell viability at >50 uM by xCELLigence system | Cricetulus griseus | 2 | ALA3217656 | cell-based format | Scientific Literature | |
| 5. | ALA3226168 | A | Cytotoxicity against Chinese hamster CHO cells overexpressing IR assessed as cell proliferation rate at 0.4 to 10 uM by xCELLigence system | Cricetulus griseus | 3 | ALA3217656 | cell-based format | Scientific Literature | |
| 6. | ALA3226169 | B | Inhibition of PTP1B in Chinese hamster CHO cells overexpressing IR assessed as insulin-stimulated IR phosphorylation treated for 3 hrs prior to insulin stimulation for 15 mins by western blot analysis | Cricetulus griseus | 3 | ALA3217656 | cell-based format | Scientific Literature | |
| 7. | ALA3226170 | B | Inhibition of human GST-tagged PTP-LAR D1D2 domain assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 3 | ALA3217656 | single protein format | Scientific Literature | |
| 8. | ALA3226171 | B | Inhibition of papaya papain assessed as Z-Phe-Arg-pNA hydrolysis by fluorometric kinetic-based assay | Carica papaya | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 9. | ALA3226172 | B | Inhibition of human GST-tagged full length MKPX assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 10. | ALA3226173 | B | Inhibition of human GST-tagged PRL2 A/S active mutant assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | assay format | Scientific Literature | |
| 11. | ALA3226174 | B | Inhibition of human GST-tagged TC-PTP catalytic domain assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 12. | ALA3226175 | B | Inhibition of human GST-tagged PTP-sigma D1D2 domain assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 13. | ALA3226176 | B | Inhibition of human GST-tagged PTP1B catalytic domain assessed as DiFMUP hydrolysis by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 14. | ALA3226177 | B | Inhibition of papaya papain assessed as Z-Phe-Arg-pNA hydrolysis at 10 uM by fluorometric kinetic-based assay | Carica papaya | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 15. | ALA3226178 | B | Inhibition of human GST-tagged full length MKPX assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 16. | ALA3226179 | B | Inhibition of human GST-tagged PRL2 A/S active mutant assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | assay format | Scientific Literature | |
| 17. | ALA3226180 | B | Inhibition of human GST-tagged PTP-LAR D1D2 domain assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 18. | ALA3226181 | B | Inhibition of human GST-tagged PTP-sigma D1D2 domain assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 19. | ALA3226182 | B | Inhibition of human GST-tagged PTP1B catalytic domain assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature | |
| 20. | ALA3226183 | B | Inhibition of human GST-tagged TC-PTP catalytic domain assessed as DiFMUP hydrolysis at 10 uM by fluorometric kinetic-based assay | Homo sapiens | 6 | ALA3217656 | single protein format | Scientific Literature |
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