| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1831365 | T | Toxicity in po dosed athymic nu/nu Harlan mouse with xenografted human HCT116 cells assessed as maximum tolerated administered qd for 7 days | Mus musculus | 1 | ALA1828590 | organism-based format | Scientific Literature | |
| 2. | ALA1832515 | B | Inhibition of full length recombinant HDAC1 using Fluor de Lys as substrate by fluorescence assay | 51 | ALA1828590 | single protein format | Scientific Literature | ||
| 3. | ALA1832516 | F | Antiproliferative activity against human COLO205 cells after 96 hrs by celltiter 96 assay | Homo sapiens | 51 | ALA1828590 | cell-based format | Scientific Literature | |
| 4. | ALA1832517 | F | Antiproliferative activity against human A2780 cells after 96 hrs by celltiter 96 assay | Homo sapiens | 20 | ALA1828590 | cell-based format | Scientific Literature | |
| 5. | ALA1832518 | F | Antiproliferative activity against human HCT116 cells after 96 hrs by celltiter 96 assay | Homo sapiens | 20 | ALA1828590 | cell-based format | Scientific Literature | |
| 6. | ALA1832519 | F | Antiproliferative activity against human PC3 cells after 96 hrs by celltiter 96 assay | Homo sapiens | 20 | ALA1828590 | cell-based format | Scientific Literature | |
| 7. | ALA1832520 | B | Competitive inhibition of HDAC1 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 8. | ALA1832521 | B | Competitive inhibition of HDAC2 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 9. | ALA1832522 | B | Competitive inhibition of HDAC3 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 10. | ALA1832523 | B | Competitive inhibition of HDAC4 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 11. | ALA1832524 | B | Competitive inhibition of HDAC5 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 12. | ALA1832525 | B | Competitive inhibition of HDAC6 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 13. | ALA1832526 | B | Competitive inhibition of HDAC7 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 14. | ALA1832527 | B | Competitive inhibition of HDAC8 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 15. | ALA1832528 | B | Competitive inhibition of HDAC9 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 16. | ALA1832529 | B | Competitive inhibition of HDAC10 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 17. | ALA1832530 | B | Competitive inhibition of HDAC11 using KI-104 as substrate by fluorescence assay | 14 | ALA1828590 | single protein format | Scientific Literature | ||
| 18. | ALA1832815 | A | Inhibition of recombinant CYP3A4 after 30 mins by fluorescence assay | 3 | ALA1828590 | single protein format | Scientific Literature | ||
| 19. | ALA1832816 | A | Inhibition of recombinant CYP2D6 after 30 mins by fluorescence assay | 3 | ALA1828590 | single protein format | Scientific Literature | ||
| 20. | ALA1832817 | A | Inhibition of CYP1A in human liver microsomes by fluorescence assay | Homo sapiens | 3 | ALA1828590 | microsome format | Scientific Literature |
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