| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1833210 | B | Inhibition of human PDE4B1 assessed as inhibition of [3H]cAMP hydrolysis to [3H]AMP after 15 mins by scintillation proximity assay | Homo sapiens | 18 | ALA1828553 | single protein format | Scientific Literature | |
| 2. | ALA1833211 | B | Inhibition of human PDE4A4 assessed as inhibition of [3H]cAMP hydrolysis to [3H]AMP after 15 mins by scintillation proximity assay | Homo sapiens | 17 | ALA1828553 | single protein format | Scientific Literature | |
| 3. | ALA1833212 | B | Inhibition of human PDE4D3 assessed as inhibition of [3H]cAMP hydrolysis to [3H]AMP after 15 mins by scintillation proximity assay | Homo sapiens | 17 | ALA1828553 | single protein format | Scientific Literature | |
| 4. | ALA1833213 | F | Inhibition of LPS-induced TNFalpha production in human whole blood after 24 hrs by ELISA | Homo sapiens | 17 | ALA1828553 | tissue-based format | Scientific Literature | |
| 5. | ALA1833214 | F | Inhibition of LPS-induced TNFalpha production in PBMC | 2 | ALA1828553 | cell-based format | Scientific Literature | ||
| 6. | ALA1833215 | F | Inhibition of LPS-induced TNFalpha production in neutrophilia rat at 0.3 mg/kg, po | Rattus norvegicus | 2 | ALA1828553 | organism-based format | Scientific Literature | |
| 7. | ALA1833216 | F | Antiemetic activity in po dosed ferret up to 3 hrs | Mustela putorius furo | 2 | ALA1828553 | organism-based format | Scientific Literature | |
| 8. | ALA1833217 | A | Metabolic stability in rat liver microsomes | Rattus norvegicus | 2 | ALA1828553 | microsome format | Scientific Literature | |
| 9. | ALA1833218 | A | Metabolic stability in human liver microsomes after 30 mins by HPLC-UV method | Homo sapiens | 2 | ALA1828553 | microsome format | Scientific Literature | |
| 10. | ALA1833219 | A | Cmax in ferret at 0.1 mg/kg, po | Mustela putorius furo | 1 | ALA1828553 | organism-based format | Scientific Literature | |
| 11. | ALA1833221 | A | Half life in ferret at 0.1 mg/kg, po | Mustela putorius furo | 1 | ALA1828553 | organism-based format | Scientific Literature | |
| 12. | ALA1833223 | A | Tmax in ferret at 0.1 mg/kg, po | Mustela putorius furo | 1 | ALA1828553 | organism-based format | Scientific Literature | |
| 13. | ALA1833225 | A | AUC (0 to t) in ferret at 0.1 mg/kg, po | Mustela putorius furo | 1 | ALA1828553 | organism-based format | Scientific Literature | |
| 14. | ALA1833227 | A | Apparent permeability across human Caco2 cells after 3 hrs | Homo sapiens | 2 | ALA1828553 | cell-based format | Scientific Literature |
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