| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1838817 | B | Displacement of [3H]AMPA from recombinant rat GluA1 flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 2. | ALA1837932 | B | Displacement of [3H]AMPA from AMPA receptor in rat brain synaptosomal membranes | Rattus norvegicus | 10 | ALA1833858 | cell membrane format | Scientific Literature | |
| 3. | ALA1837935 | B | Displacement of [3H]AMPA from recombinant rat GluA2(R) flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 4. | ALA1837936 | B | Displacement of [3H]AMPA from recombinant rat GluA3 flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 5. | ALA1837937 | B | Displacement of [3H]AMPA from recombinant rat GluA4 flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 6. | ALA1837938 | B | Displacement of [3H]AMPA from recombinant rat GluA1 receptor flop isoform Y716F mutant expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 7. | ALA1837939 | B | Displacement of [3H]AMPA from recombinant GluA2 S1S2J soluble ligand binding domain | 1 | ALA1833858 | single protein format | Scientific Literature | ||
| 8. | ALA1837940 | B | Displacement of [3H]AMPA from recombinant GluA2 S1S2J soluble ligand binding domain Y702F mutant | 1 | ALA1833858 | assay format | Scientific Literature | ||
| 9. | ALA1837941 | B | Selectivity ratio of Ki for recombinant rat GluA3 flop isoform receptor expressed in Sf9 insect cell membrane to Ki for recombinant rat GluA1 flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 10. | ALA1837942 | B | Selectivity ratio of Ki for recombinant rat GluA4 flop isoform receptor expressed in Sf9 insect cell membrane to Ki for recombinant rat GluA1 flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 11. | ALA1838450 | B | Selectivity ratio of Ki for recombinant rat GluA3 flop isoform receptor expressed in Sf9 insect cell membrane to Ki for recombinant rat GluA2(R) flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 12. | ALA1838451 | B | Selectivity ratio of Ki for recombinant rat GluA4 flop isoform receptor expressed in Sf9 insect cell membrane to Ki for recombinant rat GluA2(R) flop isoform receptor expressed in Sf9 insect cell membrane | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 13. | ALA1838452 | F | Antagonist activity at recombinant rat GluA2(Q) flip isoform receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -45 mV holding potential by two-electrode voltage clamp electrophysiology | Rattus norvegicus | 3 | ALA1833858 | cell-based format | Scientific Literature | |
| 14. | ALA1838453 | F | Antagonist activity at recombinant rat GluA3 flip isoform receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current at -90 mV holding potential by two-electrode voltage clamp electrophysiology | Rattus norvegicus | 3 | ALA1833858 | cell-based format | Scientific Literature | |
| 15. | ALA1838454 | B | Selectivity ratio of Kb for recombinant rat GluA2(Q) flip isoform receptor expressed in Xenopus laevis oocytes to Kb for recombinant rat GluA3 flip isoform receptor expressed in Xenopus laevis oocytes | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 16. | ALA1838455 | F | Competitive antagonist activity at recombinant rat GluA2(Q) flip isoform receptor expressed in Xenopus laevis oocytes assessed as maximal inhibition of glutamate-induced current at -60 mV holding potential by two-electrode voltage clamp electrophysiology | Rattus norvegicus | 1 | ALA1833858 | cell-based format | Scientific Literature | |
| 17. | ALA3379223 | B | Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation counting | Rattus norvegicus | 3 | ALA3351684 | cell-based format | Scientific Literature | |
| 18. | ALA3379751 | B | Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation counting | Rattus norvegicus | 3 | ALA3351684 | cell-based format | Scientific Literature | |
| 19. | ALA3379754 | B | Displacement of [3H]AMPA from AMPA receptor in rat brain cortex after 30 mins by Packard TopCount microplate scintillator counting | Rattus norvegicus | 18 | ALA3351684 | tissue-based format | Scientific Literature |
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